Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50055523 (CHEMBL3321792) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523091 (CHEMBL4577233) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523091 (CHEMBL4577233) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50055523 (CHEMBL3321792) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523093 (CHEMBL4446729) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523093 (CHEMBL4446729) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50363895 (CHEMBL1946126) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50363895 (CHEMBL1946126) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50363896 (CHEMBL1946253) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50363896 (CHEMBL1946253) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523678 (CHEMBL4556093) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523678 (CHEMBL4556093) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50262929 (4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluo...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523683 (CHEMBL4566049) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523683 (CHEMBL4566049) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50362857 (CHEMBL1940412) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50262929 (4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluo...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50363895 (CHEMBL1946126) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50363895 (CHEMBL1946126) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523091 (CHEMBL4577233) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523091 (CHEMBL4577233) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523096 (CHEMBL4574793) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523096 (CHEMBL4574793) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50055522 (CHEMBL3321791) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50055522 (CHEMBL3321791) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523095 (CHEMBL4573441) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523095 (CHEMBL4573441) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50363896 (CHEMBL1946253) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50363896 (CHEMBL1946253) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523092 (CHEMBL4581305) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523681 (CHEMBL4558031) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523681 (CHEMBL4558031) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50055520 (CHEMBL3321789) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50055520 (CHEMBL3321789) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523676 (CHEMBL4529943) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523684 (CHEMBL4463587) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523684 (CHEMBL4463587) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50055519 (CHEMBL3321788) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50055519 (CHEMBL3321788) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523682 (CHEMBL4474014) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523682 (CHEMBL4474014) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement of [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK293T cell membranes | Bioorg Med Chem 27: 2629-2636 (2019) Article DOI: 10.1016/j.bmc.2019.04.012 BindingDB Entry DOI: 10.7270/Q2PZ5D7G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50262929 (4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50262929 (4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523095 (CHEMBL4573441) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50523089 (CHEMBL4554850) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50362859 (CHEMBL1940414) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma intracellular receptor 2 (Homo sapiens (Human)) | BDBM50055519 (CHEMBL3321788) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-DTG from sigma 2 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50523095 (CHEMBL4573441) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A&M University Curated by ChEMBL | Assay Description Displacement [3H]-Pentazocine from sigma 1 receptor (unknown origin) expressed in HEK cell membranes | Bioorg Med Chem 27: 2421-2426 (2019) Article DOI: 10.1016/j.bmc.2019.01.035 BindingDB Entry DOI: 10.7270/Q2FJ2M62 | |||||||||||
More data for this Ligand-Target Pair |
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