Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
P-selectin (Homo sapiens (Human)) | BDBM50027066 (CHEMBL3335534) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026881 (CHEMBL3335530) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026887 (CHEMBL3335533) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026870 (CHEMBL3335528) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50400720 (CHEMBL2204272) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50400720 (CHEMBL2204272) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of immobilized rhPSGL-Ig binding to soluble P-selectin by surface plasmon resonance competitive binding assay | ACS Med Chem Lett 3: 1045-1049 (2012) Article DOI: 10.1021/ml300263x BindingDB Entry DOI: 10.7270/Q2F47Q8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026882 (CHEMBL3335531) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026886 (CHEMBL3335532) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026871 (CHEMBL3335529) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026881 (CHEMBL3335530) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
E-selectin (Homo sapiens (Human)) | BDBM50026881 (CHEMBL3335530) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026870 (CHEMBL3335528) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
E-selectin (Homo sapiens (Human)) | BDBM50026870 (CHEMBL3335528) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026871 (CHEMBL3335529) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
E-selectin (Homo sapiens (Human)) | BDBM50026871 (CHEMBL3335529) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026869 (CHEMBL3335527) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50400721 (CHEMBL2204273) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.80E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) by surface plasmon resonance-based dynamic assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50400721 (CHEMBL2204273) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.80E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of immobilized rhPSGL-Ig binding to soluble P-selectin by surface plasmon resonance competitive binding assay | ACS Med Chem Lett 3: 1045-1049 (2012) Article DOI: 10.1021/ml300263x BindingDB Entry DOI: 10.7270/Q2F47Q8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50400719 (CHEMBL2204271) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of immobilized rhPSGL-Ig binding to soluble P-selectin by surface plasmon resonance competitive binding assay | ACS Med Chem Lett 3: 1045-1049 (2012) Article DOI: 10.1021/ml300263x BindingDB Entry DOI: 10.7270/Q2F47Q8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50400722 (CHEMBL2204274) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of immobilized rhPSGL-Ig binding to soluble P-selectin by surface plasmon resonance competitive binding assay | ACS Med Chem Lett 3: 1045-1049 (2012) Article DOI: 10.1021/ml300263x BindingDB Entry DOI: 10.7270/Q2F47Q8Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50026869 (CHEMBL3335527) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
E-selectin (Homo sapiens (Human)) | BDBM50026869 (CHEMBL3335527) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.08E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P-selectin (Homo sapiens (Human)) | BDBM50400721 (CHEMBL2204273) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.84E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at P-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
E-selectin (Homo sapiens (Human)) | BDBM50400721 (CHEMBL2204273) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.46E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Cliniques de Montr£al (IRCM) Curated by ChEMBL | Assay Description Antagonist activity at E-selectin (unknown origin) assessed as adhesion to [3H]thymidine-labelled human HL60 cells by static assay | ACS Med Chem Lett 5: 1054-9 (2014) Article DOI: 10.1021/ml500266x BindingDB Entry DOI: 10.7270/Q2KW5HNG | |||||||||||
More data for this Ligand-Target Pair |