Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Nociceptin receptor
(Homo sapiens (Human)) | BDBM172401
(US9090618, ZA14 | US9598411, Ref. No. ZA14)Show SMILES C[C@H]1C[C@H]2C[C@@H](C1)C[C@@H](C2)N1[C@H]2CCC[C@@H]1C[C@@H](C2)n1c(nc2ccccc12)N1CCC[C@H]1C(O)=O |r,THB:8:10:17.18.16:12.14.13| Show InChI InChI=1S/C30H42N4O2/c1-19-12-20-14-21(13-19)16-24(15-20)33-22-6-4-7-23(33)18-25(17-22)34-27-9-3-2-8-26(27)31-30(34)32-11-5-10-28(32)29(35)36/h2-3,8-9,19-25,28H,4-7,10-18H2,1H3,(H,35,36)/t19-,20-,21+,22-,23+,24+,25+,28-/m0/s1 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
Similars
| US Patent
| 505 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue Pharma L.P.
US Patent
| Assay Description
δ-Opioid Receptor Binding Assay Procedures: Radioligand dose-displacement assays used 0.2 nM [3H]-Naltrindole (NEN; 33.0 Ci/mmole) with 10-20 &#... |
US Patent US9598411 (2017)
BindingDB Entry DOI: 10.7270/Q2ZG6V9S |
More data for this
Ligand-Target Pair | |
Opioid growth factor receptor-like protein 1
(Homo sapiens (Human)) | BDBM172401
(US9090618, ZA14 | US9598411, Ref. No. ZA14)Show SMILES C[C@H]1C[C@H]2C[C@@H](C1)C[C@@H](C2)N1[C@H]2CCC[C@@H]1C[C@@H](C2)n1c(nc2ccccc12)N1CCC[C@H]1C(O)=O |r,THB:8:10:17.18.16:12.14.13| Show InChI InChI=1S/C30H42N4O2/c1-19-12-20-14-21(13-19)16-24(15-20)33-22-6-4-7-23(33)18-25(17-22)34-27-9-3-2-8-26(27)31-30(34)32-11-5-10-28(32)29(35)36/h2-3,8-9,19-25,28H,4-7,10-18H2,1H3,(H,35,36)/t19-,20-,21+,22-,23+,24+,25+,28-/m0/s1 | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
Similars
| US Patent
| 505 | -35.9 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
Purdue Pharma L.P.
US Patent
| Assay Description
Radioligand binding assays (screening and dose-displacement) used 0.1 nM [3H]-nociceptin (NEN; 87.7 Ci/mmole) with 10-20 ug membrane protein in a fin... |
US Patent US9090618 (2015)
BindingDB Entry DOI: 10.7270/Q2G73CGB |
More data for this
Ligand-Target Pair | |