Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Cysteinyl leukotriene receptor 1
(GUINEA PIG) | BDBM50284890
((1-{(R)-1-{3-[(E)-2-(4-Cyclopropyl-thiazol-2-yl)-v...)Show SMILES CC(C)(O)c1ccccc1CC[C@@H](SCC1(CC(O)=O)CC1)c1cccc(\C=C\c2nc(cs2)C2CC2)c1 Show InChI InChI=1S/C32H37NO3S2/c1-31(2,36)26-9-4-3-7-23(26)13-14-28(38-21-32(16-17-32)19-30(34)35)25-8-5-6-22(18-25)10-15-29-33-27(20-37-29)24-11-12-24/h3-10,15,18,20,24,28,36H,11-14,16-17,19,21H2,1-2H3,(H,34,35)/b15-10+/t28-/m1/s1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Inhibition of [3H]-LTD4 binding on guinea-pig lung membranes |
Bioorg Med Chem Lett 5: 1615-1620 (1995)
Article DOI: 10.1016/0960-894X(95)00265-U
BindingDB Entry DOI: 10.7270/Q2NV9J6V |
More data for this
Ligand-Target Pair | |
Cysteinyl leukotriene receptor 1
(GUINEA PIG) | BDBM50284890
((1-{(R)-1-{3-[(E)-2-(4-Cyclopropyl-thiazol-2-yl)-v...)Show SMILES CC(C)(O)c1ccccc1CC[C@@H](SCC1(CC(O)=O)CC1)c1cccc(\C=C\c2nc(cs2)C2CC2)c1 Show InChI InChI=1S/C32H37NO3S2/c1-31(2,36)26-9-4-3-7-23(26)13-14-28(38-21-32(16-17-32)19-30(34)35)25-8-5-6-22(18-25)10-15-29-33-27(20-37-29)24-11-12-24/h3-10,15,18,20,24,28,36H,11-14,16-17,19,21H2,1-2H3,(H,34,35)/b15-10+/t28-/m1/s1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
| n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description
Inhibition of [3H]LTD4 binding on guinea-pig lung membranes |
Bioorg Med Chem Lett 5: 1615-1620 (1995)
Article DOI: 10.1016/0960-894X(95)00265-U
BindingDB Entry DOI: 10.7270/Q2NV9J6V |
More data for this
Ligand-Target Pair | |