Found 5 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Cannabinoid receptor 1
(Homo sapiens (Human)) | BDBM50398233
(CHEMBL2177253)Show InChI InChI=1S/C23H26O3/c1-4-5-6-10-17-12-21(25-3)20-15-19(23(24)26-22(20)13-17)14-18-11-8-7-9-16(18)2/h7-9,11-13,15H,4-6,10,14H2,1-3H3 | PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn
Curated by ChEMBL
| Assay Description
Displacement of [3H]CP55,940 from human CB1 receptor expressed in CHO cells after 2 hrs by liquid scintillation counter |
J Med Chem 55: 7967-77 (2012)
Article DOI: 10.1021/jm3008213
BindingDB Entry DOI: 10.7270/Q2JM2BRJ |
More data for this
Ligand-Target Pair | |
Cannabinoid receptor 2
(Homo sapiens (Human)) | BDBM50398233
(CHEMBL2177253)Show InChI InChI=1S/C23H26O3/c1-4-5-6-10-17-12-21(25-3)20-15-19(23(24)26-22(20)13-17)14-18-11-8-7-9-16(18)2/h7-9,11-13,15H,4-6,10,14H2,1-3H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 405 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn
Curated by ChEMBL
| Assay Description
Displacement of [3H]CP55,940 from human CB2 receptor expressed in CHO cells after 2 hrs by liquid scintillation counter |
J Med Chem 55: 7967-77 (2012)
Article DOI: 10.1021/jm3008213
BindingDB Entry DOI: 10.7270/Q2JM2BRJ |
More data for this
Ligand-Target Pair | |
G-protein coupled receptor 55
(Homo sapiens (Human)) | BDBM50398233
(CHEMBL2177253)Show InChI InChI=1S/C23H26O3/c1-4-5-6-10-17-12-21(25-3)20-15-19(23(24)26-22(20)13-17)14-18-11-8-7-9-16(18)2/h7-9,11-13,15H,4-6,10,14H2,1-3H3 | Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 5.08E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn
Curated by ChEMBL
| Assay Description
Antagonist activity at human GPR55 transfected in CHO cells assessed as inhibition of LPI-induced beta-arrestin recruitment incubated 60 mins prior t... |
J Med Chem 56: 4798-810 (2013)
Article DOI: 10.1021/jm4005175
BindingDB Entry DOI: 10.7270/Q2GM88QX |
More data for this
Ligand-Target Pair | |
N-arachidonyl glycine receptor
(Homo sapiens (Human)) | BDBM50398233
(CHEMBL2177253)Show InChI InChI=1S/C23H26O3/c1-4-5-6-10-17-12-21(25-3)20-15-19(23(24)26-22(20)13-17)14-18-11-8-7-9-16(18)2/h7-9,11-13,15H,4-6,10,14H2,1-3H3 | Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn
Curated by ChEMBL
| Assay Description
Antagonist activity at human GPR18 transfected in CHO cells assessed as delta9-THC-induced beta-arrestin recruitment incubated 60 mins prior to delta... |
J Med Chem 56: 4798-810 (2013)
Article DOI: 10.1021/jm4005175
BindingDB Entry DOI: 10.7270/Q2GM88QX |
More data for this
Ligand-Target Pair | |
Cannabinoid receptor 2
(Homo sapiens (Human)) | BDBM50398233
(CHEMBL2177253)Show InChI InChI=1S/C23H26O3/c1-4-5-6-10-17-12-21(25-3)20-15-19(23(24)26-22(20)13-17)14-18-11-8-7-9-16(18)2/h7-9,11-13,15H,4-6,10,14H2,1-3H3 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | n/a | n/a | 213 | n/a | n/a | n/a | n/a |
University of Bonn
Curated by ChEMBL
| Assay Description
Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation using [3H]-cAMP after ... |
J Med Chem 55: 7967-77 (2012)
Article DOI: 10.1021/jm3008213
BindingDB Entry DOI: 10.7270/Q2JM2BRJ |
More data for this
Ligand-Target Pair | |