Found 2 hits in this display Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Lysosomal Pro-X carboxypeptidase
(Homo sapiens (Human)) | BDBM193270
(US9193762, RS-33-15)Show SMILES COc1ccccc1CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 Show InChI InChI=1S/C26H31N3O5/c1-33-23-14-6-5-11-20(23)17-27-24(30)21-12-7-15-28(21)25(31)22-13-8-16-29(22)26(32)34-18-19-9-3-2-4-10-19/h2-6,9-11,14,21-22H,7-8,12-13,15-18H2,1H3,(H,27,30)/t21-,22-/m0/s1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| US Patent
| 2.89E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UNIVERSITY OF MISSISSIPPI
US Patent
| Assay Description Briefly, rPRCP was incubated in the presence or absence of various PRCP inhibitors in HEPES-carbonated buffer containing 1 mM Ala-Pro-paranitroanilin... |
US Patent US9193762 (2015)
BindingDB Entry DOI: 10.7270/Q2ST7NN2 |
More data for this Ligand-Target Pair | |
Lysosomal Pro-X carboxypeptidase
(Homo sapiens (Human)) | BDBM193270
(US9193762, RS-33-15)Show SMILES COc1ccccc1CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 Show InChI InChI=1S/C26H31N3O5/c1-33-23-14-6-5-11-20(23)17-27-24(30)21-12-7-15-28(21)25(31)22-13-8-16-29(22)26(32)34-18-19-9-3-2-4-10-19/h2-6,9-11,14,21-22H,7-8,12-13,15-18H2,1H3,(H,27,30)/t21-,22-/m0/s1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| US Patent
| 7.71E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UNIVERSITY OF MISSISSIPPI
US Patent
| Assay Description Human pulmonary artery endothelial cells (HPAEC) were purchased from Invitrogen (Carlsbad, Calif.) and were cultured as previously described.20 The c... |
US Patent US9193762 (2015)
BindingDB Entry DOI: 10.7270/Q2ST7NN2 |
More data for this Ligand-Target Pair | |