Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Alpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase
(Homo sapiens (Human)) | BDBM235206
(US9365558, 29 | US9822074, 29)Show SMILES Cc1ccc(cc1)C1=C(C(=O)NS(=O)(=O)c2ccccc2)C(=O)N[C@@](C1)(c1ccc(OCCCC(F)(F)F)cc1)C(F)(F)F |r,c:8| Show InChI InChI=1S/C30H26F6N2O5S/c1-19-8-10-20(11-9-19)24-18-28(30(34,35)36,21-12-14-22(15-13-21)43-17-5-16-29(31,32)33)37-26(39)25(24)27(40)38-44(41,42)23-6-3-2-4-7-23/h2-4,6-15H,5,16-18H2,1H3,(H,37,39)(H,38,40)/t28-/m0/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 84 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The MGAT enzyme reactions were performed in Corning FALCONŽ 96-well Polypropylene plates, in a total volume of 60 μL of 50 mM Potassium Phosphat... |
US Patent US9822074 (2017)
BindingDB Entry DOI: 10.7270/Q2K939TM |
More data for this
Ligand-Target Pair | |
Alpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase
(Homo sapiens (Human)) | BDBM235206
(US9365558, 29 | US9822074, 29)Show SMILES Cc1ccc(cc1)C1=C(C(=O)NS(=O)(=O)c2ccccc2)C(=O)N[C@@](C1)(c1ccc(OCCCC(F)(F)F)cc1)C(F)(F)F |r,c:8| Show InChI InChI=1S/C30H26F6N2O5S/c1-19-8-10-20(11-9-19)24-18-28(30(34,35)36,21-12-14-22(15-13-21)43-17-5-16-29(31,32)33)37-26(39)25(24)27(40)38-44(41,42)23-6-3-2-4-7-23/h2-4,6-15H,5,16-18H2,1H3,(H,37,39)(H,38,40)/t28-/m0/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 84 | n/a | n/a | n/a | n/a | 7.4 | 65 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The MGAT enzyme reactions were performed in Corning FALCON® 96-well Polypropylene plates, in a total volume of 60 μL of 50 mM Potassium Phosph... |
US Patent US9365558 (2016)
BindingDB Entry DOI: 10.7270/Q2XS5T8B |
More data for this
Ligand-Target Pair | |