Found 3 hits in this display Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Alpha-1D adrenergic receptor
(Homo sapiens (Human)) | BDBM50000202
(CHEMBL142958)Show InChI InChI=1S/C15H16N2OS/c1-11-6-7-14(19-11)12-4-2-3-5-13(12)18-10-15-16-8-9-17-15/h2-7H,8-10H2,1H3,(H,16,17) | Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | n/a | n/a | <1.00E+5 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Research and Development
Curated by ChEMBL
| Assay Description Activation of recombinant human adrenergic, alpha-1D receptor expressed in rat-1 fibroblasts assayed via calcium mobilization through Gq coupled PLC ... |
Bioorg Med Chem Lett 12: 471-5 (2002)
Checked by Author BindingDB Entry DOI: 10.7270/Q22V2HD6 |
More data for this Ligand-Target Pair | |
Alpha-1B adrenergic receptor
(Homo sapiens (Human)) | BDBM50000202
(CHEMBL142958)Show InChI InChI=1S/C15H16N2OS/c1-11-6-7-14(19-11)12-4-2-3-5-13(12)18-10-15-16-8-9-17-15/h2-7H,8-10H2,1H3,(H,16,17) | UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | n/a | n/a | <1.00E+5 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Research and Development
Curated by ChEMBL
| Assay Description Activation of recombinant human adrenergic, alpha-1B receptor expressed in rat-1 fibroblasts determined via calcium mobilization through Gq coupled P... |
Bioorg Med Chem Lett 12: 471-5 (2002)
Checked by Author BindingDB Entry DOI: 10.7270/Q22V2HD6 |
More data for this Ligand-Target Pair | |
Alpha-1A adrenergic receptor
(Homo sapiens (Human)) | BDBM50000202
(CHEMBL142958)Show InChI InChI=1S/C15H16N2OS/c1-11-6-7-14(19-11)12-4-2-3-5-13(12)18-10-15-16-8-9-17-15/h2-7H,8-10H2,1H3,(H,16,17) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Research and Development
Curated by ChEMBL
| Assay Description Activation of recombinant human adrenergic,alpha-1A receptor expressed in rat-1 fibroblasts determined via calcium mobilization through Gq coupled PL... |
Bioorg Med Chem Lett 12: 471-5 (2002)
Checked by Author BindingDB Entry DOI: 10.7270/Q22V2HD6 |
More data for this Ligand-Target Pair | |