Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Neutral amino acid transporter B(0)
(Homo sapiens (Human)) | BDBM464424
(US10793514, Compound 17)Show SMILES Cc1cccc(COc2ccccc2CN(CC[C@@H](N)C(O)=O)Cc2ccccc2OCc2cccc(C)c2)c1 |r| Show InChI InChI=1S/C34H38N2O4/c1-25-9-7-11-27(19-25)23-39-32-15-5-3-13-29(32)21-36(18-17-31(35)34(37)38)22-30-14-4-6-16-33(30)40-24-28-12-8-10-26(2)20-28/h3-16,19-20,31H,17-18,21-24,35H2,1-2H3,(H,37,38)/t31-/m1/s1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet 
| Purchase
PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University
US Patent
| Assay Description
Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... |
US Patent US10793514 (2020)
BindingDB Entry DOI: 10.7270/Q2TT4V1N |
More data for this
Ligand-Target Pair | |
Amino acid transporter
(Rattus norvegicus) | BDBM464424
(US10793514, Compound 17)Show SMILES Cc1cccc(COc2ccccc2CN(CC[C@@H](N)C(O)=O)Cc2ccccc2OCc2cccc(C)c2)c1 |r| Show InChI InChI=1S/C34H38N2O4/c1-25-9-7-11-27(19-25)23-39-32-15-5-3-13-29(32)21-36(18-17-31(35)34(37)38)22-30-14-4-6-16-33(30)40-24-28-12-8-10-26(2)20-28/h3-16,19-20,31H,17-18,21-24,35H2,1-2H3,(H,37,38)/t31-/m1/s1 | UniProtKB/TrEMBL
GoogleScholar
AffyNet
| Purchase
PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 9.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University
US Patent
| Assay Description
Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... |
US Patent US10793514 (2020)
BindingDB Entry DOI: 10.7270/Q2TT4V1N |
More data for this
Ligand-Target Pair | |