Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Casein kinase I isoform delta
(Homo sapiens (Human)) | BDBM274749
(N-(6-(4-(4-fluorophenyl)-1,2- dimethyl-1H-imidazol...)Show SMILES Cc1nc(c(-c2ccc3nc(NC(=O)c4cccc(c4)-c4cccnc4)cn3n2)n1C)-c1ccc(F)cc1 Show InChI InChI=1S/C29H22FN7O/c1-18-32-27(19-8-10-23(30)11-9-19)28(36(18)2)24-12-13-26-33-25(17-37(26)35-24)34-29(38)21-6-3-5-20(15-21)22-7-4-14-31-16-22/h3-17H,1-2H3,(H,34,38) | PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 0.323 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |
Casein kinase I isoform epsilon
(Homo sapiens (Human)) | BDBM274749
(N-(6-(4-(4-fluorophenyl)-1,2- dimethyl-1H-imidazol...)Show SMILES Cc1nc(c(-c2ccc3nc(NC(=O)c4cccc(c4)-c4cccnc4)cn3n2)n1C)-c1ccc(F)cc1 Show InChI InChI=1S/C29H22FN7O/c1-18-32-27(19-8-10-23(30)11-9-19)28(36(18)2)24-12-13-26-33-25(17-37(26)35-24)34-29(38)21-6-3-5-20(15-21)22-7-4-14-31-16-22/h3-17H,1-2H3,(H,34,38) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 1.44 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |