Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Nociceptin receptor
(Homo sapiens (Human)) | BDBM172415
(US9090618, ZA38 | US9598411, Ref. No. ZA38)Show SMILES Cc1noc(C)c1S(=O)(=O)N1CCC[C@@H]1c1nc2ccccc2n1[C@@H]1C[C@@H]2CCC[C@H](C1)N2[C@H]1C[C@@H]2C[C@H](C1)CCCC2 |r,THB:33:32:24.25.31:27.29.28| Show InChI InChI=1S/C34H47N5O3S/c1-22-33(23(2)42-36-22)43(40,41)37-16-8-15-32(37)34-35-30-13-5-6-14-31(30)39(34)29-20-26-11-7-12-27(21-29)38(26)28-18-24-9-3-4-10-25(17-24)19-28/h5-6,13-14,24-29,32H,3-4,7-12,15-21H2,1-2H3/t24-,25+,26-,27+,28-,29+,32-/m1/s1 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| 780 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue Pharma L.P.
US Patent
| Assay Description
δ-Opioid Receptor Binding Assay Procedures: Radioligand dose-displacement assays used 0.2 nM [3H]-Naltrindole (NEN; 33.0 Ci/mmole) with 10-20 &#... |
US Patent US9598411 (2017)
BindingDB Entry DOI: 10.7270/Q2ZG6V9S |
More data for this
Ligand-Target Pair | |
Opioid growth factor receptor-like protein 1
(Homo sapiens (Human)) | BDBM172415
(US9090618, ZA38 | US9598411, Ref. No. ZA38)Show SMILES Cc1noc(C)c1S(=O)(=O)N1CCC[C@@H]1c1nc2ccccc2n1[C@@H]1C[C@@H]2CCC[C@H](C1)N2[C@H]1C[C@@H]2C[C@H](C1)CCCC2 |r,THB:33:32:24.25.31:27.29.28| Show InChI InChI=1S/C34H47N5O3S/c1-22-33(23(2)42-36-22)43(40,41)37-16-8-15-32(37)34-35-30-13-5-6-14-31(30)39(34)29-20-26-11-7-12-27(21-29)38(26)28-18-24-9-3-4-10-25(17-24)19-28/h5-6,13-14,24-29,32H,3-4,7-12,15-21H2,1-2H3/t24-,25+,26-,27+,28-,29+,32-/m1/s1 | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| 780 | -34.9 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
Purdue Pharma L.P.
US Patent
| Assay Description
Radioligand binding assays (screening and dose-displacement) used 0.1 nM [3H]-nociceptin (NEN; 87.7 Ci/mmole) with 10-20 ug membrane protein in a fin... |
US Patent US9090618 (2015)
BindingDB Entry DOI: 10.7270/Q2G73CGB |
More data for this
Ligand-Target Pair | |