Found 2 hits in this display Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Lysosomal Pro-X carboxypeptidase
(Homo sapiens (Human)) | BDBM193282
(US9193762, RS-37-01)Show SMILES Clc1ccccc1CNC(=O)CCCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 |r| Show InChI InChI=1S/C24H28ClN3O4/c25-20-11-5-4-10-19(20)16-27-22(29)13-6-14-26-23(30)21-12-7-15-28(21)24(31)32-17-18-8-2-1-3-9-18/h1-5,8-11,21H,6-7,12-17H2,(H,26,30)(H,27,29)/t21-/m0/s1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| US Patent
| 3.32E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UNIVERSITY OF MISSISSIPPI
US Patent
| Assay Description Briefly, rPRCP was incubated in the presence or absence of various PRCP inhibitors in HEPES-carbonated buffer containing 1 mM Ala-Pro-paranitroanilin... |
US Patent US9193762 (2015)
BindingDB Entry DOI: 10.7270/Q2ST7NN2 |
More data for this Ligand-Target Pair | |
Lysosomal Pro-X carboxypeptidase
(Homo sapiens (Human)) | BDBM193282
(US9193762, RS-37-01)Show SMILES Clc1ccccc1CNC(=O)CCCNC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 |r| Show InChI InChI=1S/C24H28ClN3O4/c25-20-11-5-4-10-19(20)16-27-22(29)13-6-14-26-23(30)21-12-7-15-28(21)24(31)32-17-18-8-2-1-3-9-18/h1-5,8-11,21H,6-7,12-17H2,(H,26,30)(H,27,29)/t21-/m0/s1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| US Patent
| 6.94E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UNIVERSITY OF MISSISSIPPI
US Patent
| Assay Description Human pulmonary artery endothelial cells (HPAEC) were purchased from Invitrogen (Carlsbad, Calif.) and were cultured as previously described.20 The c... |
US Patent US9193762 (2015)
BindingDB Entry DOI: 10.7270/Q2ST7NN2 |
More data for this Ligand-Target Pair | |