Found 2 hits in this display Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Lysosomal Pro-X carboxypeptidase
(Homo sapiens (Human)) | BDBM193266
(US9193762, RS-33-11)Show SMILES FC(F)(F)c1ccccc1CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 Show InChI InChI=1S/C26H28F3N3O4/c27-26(28,29)20-11-5-4-10-19(20)16-30-23(33)21-12-6-14-31(21)24(34)22-13-7-15-32(22)25(35)36-17-18-8-2-1-3-9-18/h1-5,8-11,21-22H,6-7,12-17H2,(H,30,33)/t21-,22-/m0/s1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| US Patent
| 1.35E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UNIVERSITY OF MISSISSIPPI
US Patent
| Assay Description Briefly, rPRCP was incubated in the presence or absence of various PRCP inhibitors in HEPES-carbonated buffer containing 1 mM Ala-Pro-paranitroanilin... |
US Patent US9193762 (2015)
BindingDB Entry DOI: 10.7270/Q2ST7NN2 |
More data for this Ligand-Target Pair | |
Lysosomal Pro-X carboxypeptidase
(Homo sapiens (Human)) | BDBM193266
(US9193762, RS-33-11)Show SMILES FC(F)(F)c1ccccc1CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1 Show InChI InChI=1S/C26H28F3N3O4/c27-26(28,29)20-11-5-4-10-19(20)16-30-23(33)21-12-6-14-31(21)24(34)22-13-7-15-32(22)25(35)36-17-18-8-2-1-3-9-18/h1-5,8-11,21-22H,6-7,12-17H2,(H,30,33)/t21-,22-/m0/s1 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| US Patent
| 4.89E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UNIVERSITY OF MISSISSIPPI
US Patent
| Assay Description Human pulmonary artery endothelial cells (HPAEC) were purchased from Invitrogen (Carlsbad, Calif.) and were cultured as previously described.20 The c... |
US Patent US9193762 (2015)
BindingDB Entry DOI: 10.7270/Q2ST7NN2 |
More data for this Ligand-Target Pair | |