Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Casein kinase I isoform delta
(Homo sapiens (Human)) | BDBM274856
(2,6-Difluoro-N-(6-(4- (4-fluorophenyl)-1- (tetrahy...)Show SMILES Fc1ccc(cc1)-c1ncn(C2CCOCC2)c1-c1ccc2nc(NC(=O)c3cc(F)nc(F)c3)cn2n1 Show InChI InChI=1S/C26H20F3N7O2/c27-17-3-1-15(2-4-17)24-25(35(14-30-24)18-7-9-38-10-8-18)19-5-6-23-32-22(13-36(23)34-19)33-26(37)16-11-20(28)31-21(29)12-16/h1-6,11-14,18H,7-10H2,(H,33,37) | PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |
Casein kinase I isoform epsilon
(Homo sapiens (Human)) | BDBM274856
(2,6-Difluoro-N-(6-(4- (4-fluorophenyl)-1- (tetrahy...)Show SMILES Fc1ccc(cc1)-c1ncn(C2CCOCC2)c1-c1ccc2nc(NC(=O)c3cc(F)nc(F)c3)cn2n1 Show InChI InChI=1S/C26H20F3N7O2/c27-17-3-1-15(2-4-17)24-25(35(14-30-24)18-7-9-38-10-8-18)19-5-6-23-32-22(13-36(23)34-19)33-26(37)16-11-20(28)31-21(29)12-16/h1-6,11-14,18H,7-10H2,(H,33,37) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |