Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Metabotropic glutamate receptor 3
(Rattus norvegicus (Rat)) | BDBM193377
(2-(4-(((5-(4-fluorophenyl)-4-oxo-4,5,6,7-tetrahydr...)Show SMILES Fc1ccc(cc1)N1CCn2nc(CNc3ccc(cc3)C#C)cc2C1=O Show InChI InChI=1S/C21H17FN4O/c1-2-15-3-7-17(8-4-15)23-14-18-13-20-21(27)25(11-12-26(20)24-18)19-9-5-16(22)6-10-19/h1,3-10,13,23H,11-12,14H2 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 890 | n/a | n/a | n/a | n/a | n/a | 25 |
Vanderbilt University
US Patent
| Assay Description
HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m... |
US Patent US9676782 (2017)
BindingDB Entry DOI: 10.7270/Q2B8569W |
More data for this
Ligand-Target Pair | |
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat)) | BDBM193377
(2-(4-(((5-(4-fluorophenyl)-4-oxo-4,5,6,7-tetrahydr...)Show SMILES Fc1ccc(cc1)N1CCn2nc(CNc3ccc(cc3)C#C)cc2C1=O Show InChI InChI=1S/C21H17FN4O/c1-2-15-3-7-17(8-4-15)23-14-18-13-20-21(27)25(11-12-26(20)24-18)19-9-5-16(22)6-10-19/h1,3-10,13,23H,11-12,14H2 | PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | 25 |
Vanderbilt University
US Patent
| Assay Description
Gα15/TREx cells stably expressing rat mGlu3 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of a... |
US Patent US9676782 (2017)
BindingDB Entry DOI: 10.7270/Q2B8569W |
More data for this
Ligand-Target Pair | |