Found 4 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human)) | BDBM50111193
((R)-3-(1H-Indol-3-yl)-2-[(naphthalen-2-ylmethyl)-a...)Show SMILES NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NCc1ccc2ccccc2c1 Show InChI InChI=1S/C22H21N3O/c23-22(26)21(12-18-14-25-20-8-4-3-7-19(18)20)24-13-15-9-10-16-5-1-2-6-17(16)11-15/h1-11,14,21,24-25H,12-13H2,(H2,23,26)/t21-/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University
Curated by ChEMBL
| Assay Description
Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptor |
Bioorg Med Chem Lett 12: 1039-42 (2002)
BindingDB Entry DOI: 10.7270/Q2833SKD |
More data for this
Ligand-Target Pair | |
Melanocortin receptor 5
(Homo sapiens (Human)) | BDBM50111193
((R)-3-(1H-Indol-3-yl)-2-[(naphthalen-2-ylmethyl)-a...)Show SMILES NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NCc1ccc2ccccc2c1 Show InChI InChI=1S/C22H21N3O/c23-22(26)21(12-18-14-25-20-8-4-3-7-19(18)20)24-13-15-9-10-16-5-1-2-6-17(16)11-15/h1-11,14,21,24-25H,12-13H2,(H2,23,26)/t21-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 3.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University
Curated by ChEMBL
| Assay Description
Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptor |
Bioorg Med Chem Lett 12: 1039-42 (2002)
BindingDB Entry DOI: 10.7270/Q2833SKD |
More data for this
Ligand-Target Pair | |
Melanocortin receptor 3
(Homo sapiens (Human)) | BDBM50111193
((R)-3-(1H-Indol-3-yl)-2-[(naphthalen-2-ylmethyl)-a...)Show SMILES NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NCc1ccc2ccccc2c1 Show InChI InChI=1S/C22H21N3O/c23-22(26)21(12-18-14-25-20-8-4-3-7-19(18)20)24-13-15-9-10-16-5-1-2-6-17(16)11-15/h1-11,14,21,24-25H,12-13H2,(H2,23,26)/t21-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 5.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University
Curated by ChEMBL
| Assay Description
Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 3 receptor |
Bioorg Med Chem Lett 12: 1039-42 (2002)
BindingDB Entry DOI: 10.7270/Q2833SKD |
More data for this
Ligand-Target Pair | |
Melanocortin receptor 4
(Homo sapiens (Human)) | BDBM50111193
((R)-3-(1H-Indol-3-yl)-2-[(naphthalen-2-ylmethyl)-a...)Show SMILES NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NCc1ccc2ccccc2c1 Show InChI InChI=1S/C22H21N3O/c23-22(26)21(12-18-14-25-20-8-4-3-7-19(18)20)24-13-15-9-10-16-5-1-2-6-17(16)11-15/h1-11,14,21,24-25H,12-13H2,(H2,23,26)/t21-/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| 6.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University
Curated by ChEMBL
| Assay Description
Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptor |
Bioorg Med Chem Lett 12: 1039-42 (2002)
BindingDB Entry DOI: 10.7270/Q2833SKD |
More data for this
Ligand-Target Pair | |