Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Casein kinase I isoform delta
(Homo sapiens (Human)) | BDBM302486
(2-(3-Fluorophenyl)-N5- (naphthalen-1-yl)-6,7- dihy...)Show SMILES NC(=O)c1c2CN(CCn2nc1-c1cccc(F)c1)C(=O)Nc1cccc2ccccc12 Show InChI InChI=1S/C24H20FN5O2/c25-17-8-3-7-16(13-17)22-21(23(26)31)20-14-29(11-12-30(20)28-22)24(32)27-19-10-4-6-15-5-1-2-9-18(15)19/h1-10,13H,11-12,14H2,(H2,26,31)(H,27,32) | PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9598423 (2017)
BindingDB Entry DOI: 10.7270/Q2FJ2JT9 |
More data for this
Ligand-Target Pair | |
Casein kinase I isoform epsilon
(Homo sapiens (Human)) | BDBM302486
(2-(3-Fluorophenyl)-N5- (naphthalen-1-yl)-6,7- dihy...)Show SMILES NC(=O)c1c2CN(CCn2nc1-c1cccc(F)c1)C(=O)Nc1cccc2ccccc12 Show InChI InChI=1S/C24H20FN5O2/c25-17-8-3-7-16(13-17)22-21(23(26)31)20-14-29(11-12-30(20)28-22)24(32)27-19-10-4-6-15-5-1-2-9-18(15)19/h1-10,13H,11-12,14H2,(H2,26,31)(H,27,32) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9598423 (2017)
BindingDB Entry DOI: 10.7270/Q2FJ2JT9 |
More data for this
Ligand-Target Pair | |