Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Casein kinase I isoform delta
(Homo sapiens (Human)) | BDBM274649
(N-(6-amino-2-(4-fluorophenyl)- [3,6'-biimidazo[1,2...)Show SMILES Nc1ccc2nc(c(-c3ccc4nc(NC(=O)c5ccncc5)cn4n3)n2n1)-c1ccc(F)cc1 Show InChI InChI=1S/C24H16FN9O/c25-16-3-1-14(2-4-16)22-23(34-21(30-22)8-6-18(26)32-34)17-5-7-20-28-19(13-33(20)31-17)29-24(35)15-9-11-27-12-10-15/h1-13H,(H2,26,32)(H,29,35) | PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 0.694 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |
Casein kinase I isoform epsilon
(Homo sapiens (Human)) | BDBM274649
(N-(6-amino-2-(4-fluorophenyl)- [3,6'-biimidazo[1,2...)Show SMILES Nc1ccc2nc(c(-c3ccc4nc(NC(=O)c5ccncc5)cn4n3)n2n1)-c1ccc(F)cc1 Show InChI InChI=1S/C24H16FN9O/c25-16-3-1-14(2-4-16)22-23(34-21(30-22)8-6-18(26)32-34)17-5-7-20-28-19(13-33(20)31-17)29-24(35)15-9-11-27-12-10-15/h1-13H,(H2,26,32)(H,29,35) | PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| US Patent
| n/a | n/a | 2.81 | n/a | n/a | n/a | n/a | 7.4 | 25 |
Bristol-Myers Squibb Company
US Patent
| Assay Description
The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst... |
US Patent US9556179 (2017)
BindingDB Entry DOI: 10.7270/Q2G73GR5 |
More data for this
Ligand-Target Pair | |