Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Nociceptin receptor
(Homo sapiens (Human)) | BDBM172424
(US9090618, ZA47 | US9598411, Ref. No. ZA47)Show SMILES OC(=O)CCN1CCC[C@@H](Cc2nc3ccccc3n2[C@@H]2C[C@@H]3CCC[C@H](C2)N3[C@H]2C[C@@H]3C[C@H](C2)CCCC3)C1 |r,THB:29:28:20.21.27:23.25.24| Show InChI InChI=1S/C34H50N4O2/c39-34(40)14-16-36-15-6-9-26(23-36)20-33-35-31-12-3-4-13-32(31)38(33)30-21-27-10-5-11-28(22-30)37(27)29-18-24-7-1-2-8-25(17-24)19-29/h3-4,12-13,24-30H,1-2,5-11,14-23H2,(H,39,40)/t24-,25+,26-,27-,28+,29-,30+/m0/s1 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
Similars
| US Patent
| 117 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue Pharma L.P.
US Patent
| Assay Description
δ-Opioid Receptor Binding Assay Procedures: Radioligand dose-displacement assays used 0.2 nM [3H]-Naltrindole (NEN; 33.0 Ci/mmole) with 10-20 &#... |
US Patent US9598411 (2017)
BindingDB Entry DOI: 10.7270/Q2ZG6V9S |
More data for this
Ligand-Target Pair | |
Opioid growth factor receptor-like protein 1
(Homo sapiens (Human)) | BDBM172424
(US9090618, ZA47 | US9598411, Ref. No. ZA47)Show SMILES OC(=O)CCN1CCC[C@@H](Cc2nc3ccccc3n2[C@@H]2C[C@@H]3CCC[C@H](C2)N3[C@H]2C[C@@H]3C[C@H](C2)CCCC3)C1 |r,THB:29:28:20.21.27:23.25.24| Show InChI InChI=1S/C34H50N4O2/c39-34(40)14-16-36-15-6-9-26(23-36)20-33-35-31-12-3-4-13-32(31)38(33)30-21-27-10-5-11-28(22-30)37(27)29-18-24-7-1-2-8-25(17-24)19-29/h3-4,12-13,24-30H,1-2,5-11,14-23H2,(H,39,40)/t24-,25+,26-,27-,28+,29-,30+/m0/s1 | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
Similars
| US Patent
| 117 | -39.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
Purdue Pharma L.P.
US Patent
| Assay Description
Radioligand binding assays (screening and dose-displacement) used 0.1 nM [3H]-nociceptin (NEN; 87.7 Ci/mmole) with 10-20 ug membrane protein in a fin... |
US Patent US9090618 (2015)
BindingDB Entry DOI: 10.7270/Q2G73CGB |
More data for this
Ligand-Target Pair | |