Found 2 hits in this display Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Nociceptin receptor
(Homo sapiens (Human)) | BDBM172379
(US9090618, E56c(ii) | US9598411, Ref. No. E56c(ii))Show SMILES OC(=O)CN1CCCC[C@@H]1c1nc2ccccc2n1[C@@H]1C[C@@H]2CCC[C@H](C1)N2C1CCCCCCCCC1 |r,THB:28:27:19.20.26:22.24.23| Show InChI InChI=1S/C32H48N4O2/c37-31(38)23-34-20-11-10-19-30(34)32-33-28-17-8-9-18-29(28)36(32)27-21-25-15-12-16-26(22-27)35(25)24-13-6-4-2-1-3-5-7-14-24/h8-9,17-18,24-27,30H,1-7,10-16,19-23H2,(H,37,38)/t25-,26+,27+,30-/m1/s1 | PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
Similars
| US Patent
| 583 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Purdue Pharma L.P.
US Patent
| Assay Description
δ-Opioid Receptor Binding Assay Procedures: Radioligand dose-displacement assays used 0.2 nM [3H]-Naltrindole (NEN; 33.0 Ci/mmole) with 10-20 &#... |
US Patent US9598411 (2017)
BindingDB Entry DOI: 10.7270/Q2ZG6V9S |
More data for this
Ligand-Target Pair | |
Opioid growth factor receptor-like protein 1
(Homo sapiens (Human)) | BDBM172379
(US9090618, E56c(ii) | US9598411, Ref. No. E56c(ii))Show SMILES OC(=O)CN1CCCC[C@@H]1c1nc2ccccc2n1[C@@H]1C[C@@H]2CCC[C@H](C1)N2C1CCCCCCCCC1 |r,THB:28:27:19.20.26:22.24.23| Show InChI InChI=1S/C32H48N4O2/c37-31(38)23-34-20-11-10-19-30(34)32-33-28-17-8-9-18-29(28)36(32)27-21-25-15-12-16-26(22-27)35(25)24-13-6-4-2-1-3-5-7-14-24/h8-9,17-18,24-27,30H,1-7,10-16,19-23H2,(H,37,38)/t25-,26+,27+,30-/m1/s1 | KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
Similars
| US Patent
| 583 | -35.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 25 |
Purdue Pharma L.P.
US Patent
| Assay Description
Radioligand binding assays (screening and dose-displacement) used 0.1 nM [3H]-nociceptin (NEN; 87.7 Ci/mmole) with 10-20 ug membrane protein in a fin... |
US Patent US9090618 (2015)
BindingDB Entry DOI: 10.7270/Q2G73CGB |
More data for this
Ligand-Target Pair | |