Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145177 (CHEMBL3764956) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.48E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145193 (CHEMBL3765505) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145178 (CHEMBL3764721) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145189 (CHEMBL3764217) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.55E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145194 (CHEMBL3765178) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145192 (CHEMBL3765653) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145187 (CHEMBL3763533) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145184 (CHEMBL3764562) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145181 (CHEMBL3765814) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145180 (CHEMBL3763273) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145179 (CHEMBL3764020) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145195 (CHEMBL3765143) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK1/Cyclin B (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145176 ((+)-Madindoline A | CHEMBL382330) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145196 (CHEMBL3765446) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK1/Cyclin B (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50145190 (CHEMBL3763626) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Dongguk University-Seoul Curated by ChEMBL | Assay Description Inhibition of CDK2/Cyclin E (unknown origin) expressed in baculoviral infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3... | Bioorg Med Chem Lett 26: 1282-6 (2016) Article DOI: 10.1016/j.bmcl.2016.01.016 BindingDB Entry DOI: 10.7270/Q2XD13JX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50552020 (CHEMBL4777424) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to immobilized GP130 (unknown origin) by SPR analysis | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112375 BindingDB Entry DOI: 10.7270/Q27948B6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50496302 (MADINDOLINE A) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.88E+5 | n/a | n/a | n/a | n/a | n/a |
The Ohio State University Curated by ChEMBL | Assay Description Binding affinity to GP130 (unknown origin) by surface plasmon resonance analysis | J Med Chem 57: 632-41 (2014) Article DOI: 10.1021/jm401144z BindingDB Entry DOI: 10.7270/Q2B27Z87 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Interleukin-6 receptor subunit beta (Homo sapiens (Human)) | BDBM50552019 (CHEMBL4740172) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.43E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to immobilized GP130 (unknown origin) by SPR analysis | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112375 BindingDB Entry DOI: 10.7270/Q27948B6 | |||||||||||
More data for this Ligand-Target Pair |