Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteasome assembly chaperone 1/2 (Homo sapiens) | BDBM50520988![]() (CHEMBL4435319) | MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet ![]() | MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Tohoku University Curated by ChEMBL | Assay Description Inhibition of PAC1/PAC2 heterodimer (unknown origin) protein-protein interaction | Bioorg Med Chem 26: 6023-6034 (2018) Article DOI: 10.1016/j.bmc.2018.11.001 BindingDB Entry DOI: 10.7270/Q24X5C69 | |||||||||||
More data for this Ligand-Target Pair |