Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
TSC22 domain family protein 3 (Human) | BDBM476583 (US10869929, Compound 18 | US11554172, Compound 18) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476584 (US10869929, Compound 19) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM50354849 (CCI-18781 | Cutivate | FLUTICASONE PROPIONATE | Fl...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 0.150 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476575 (US10869929, Compound 8 | US11554172, Compound 8) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.25 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476572 (US10869929, Compound 6 | US11554172, Compound 6) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.320 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476567 (US10869929, Compound 3 | US11554172, Compound 3) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.440 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476573 (US10869929, Compound 7 | US11554172, Compound 7) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.450 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476568 (US10869929, Compound 4 | US11554172, Compound 4) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.710 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM50354850 (BUDESONIDE | US10869929, Compound Budesonide | US1...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476576 (US10869929, Compound 9 | US11554172, Compound 9) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.67 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476577 (US10869929, Compound 10 | US11554172, Compound 10) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.99 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476585 (US10869929, Compound 27 | US11554172, Compound 27) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM18207 ((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476591 (US10869929, Compound 30 | US11554172, Compound 30) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476593 (US10869929, Compound 31 | US11554172, Compound 31) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476589 (US10869929, Compound 28 | US11554172, Compound 28) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476581 (US10869929, Compound 14 | US11554172, Compound 14) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18.1 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476590 (US10869929, Compound 29 | US11554172, Compound 29) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 24.2 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476594 (US10869929, Compound 32 | US11554172, Compound 32) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 115 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476569 (US10869929, Compound 5 | US11554172, Compound 5) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476579 (US10869929, Compound 12 | US11554172, Compound 12) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 162 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
TSC22 domain family protein 3 (Human) | BDBM476580 (US10869929, Compound 13 | US11554172, Compound 13) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
MERCK SHARP & DOHME CORP. US Patent | Assay Description HUT78 cells were cultured in IMEM plus 20% heat inactivated FBS and cell density was maintained between 0.1 to 1.2 million/mL. 786-O cells were cultu... | US Patent US10869929 (2020) BindingDB Entry DOI: 10.7270/Q2N58QG7 | |||||||||||
More data for this Ligand-Target Pair |