Found 102 hits Enz. Inhib. hit(s) with Target = 'Transcriptional enhancer factor TEF-5' Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626326
(7-(4-isopropylphenyl)-5-[(2- methylene-3-oxo-buty...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(C)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet 
| PC cid
PC sid
UniChem
| | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626323
(US11787775, Compound 8 | methyl 2-[[[4-cyano-7-(4-...)Show SMILES COC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)C(C)C | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626354
(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626354
(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626324
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 430 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626350
(2-[[[4-cyano-7-(4-isopropyl-2- thienyl)-2,3-dihyd...)Show SMILES CC(C)c1csc(c1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 430 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626362
(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)Show SMILES OCc1c2CCOc2c(cc1NCC(=C)C(=O)NO)-c1ccc(OC(F)(F)F)cc1 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626362
(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)Show SMILES OCc1c2CCOc2c(cc1NCC(=C)C(=O)NO)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626358
(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)Show SMILES ONC(=O)C(=C)CNc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncsc2c1C#N | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 660 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626318
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626354
(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626354
(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 710 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626355
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 710 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626324
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 850 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626361
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES OC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 920 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626355
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES ONC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 970 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626340
(2-[[[6-cyano-5-[(E)-2-[trans-4- (trifluoromethyl)...)Show SMILES OC(=O)C(=C)CNc1cnc(C#N)c(\C=C\[C@H]2CC[C@@H](CC2)C(F)(F)F)c1 |r,wU:16.15,wD:19.22,(-8.67,1.15,;-7.34,1.93,;-7.34,3.47,;-6,1.15,;-6,-.38,;-4.67,1.93,;-3.33,1.15,;-2,1.93,;-2,3.47,;-.67,4.23,;.67,3.47,;2,4.23,;3.33,5,;.67,1.93,;2,1.15,;2,-.38,;3.33,-1.15,;4.67,-.38,;6,-1.15,;6,-2.69,;4.67,-3.47,;3.33,-2.69,;7.34,-3.47,;8.67,-2.69,;7.34,-5,;8.67,-4.23,;-.67,1.15,)| | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 970 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626350
(2-[[[4-cyano-7-(4-isopropyl-2- thienyl)-2,3-dihyd...)Show SMILES CC(C)c1csc(c1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626365
(2-[[[7-cyano-4-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES ONC(=O)C(=C)CNc1cc(-c2ccc(cc2)S(F)(F)(F)(F)F)c2ncsc2c1C#N | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626360
(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626339
(2-[[[6-methoxy-5-[(E)-2-[trans-4- (trifluoromethy...)Show SMILES COc1ncc(NCC(=C)C(O)=O)cc1\C=C\[C@H]1CC[C@@H](CC1)C(F)(F)F |r,wU:17.17,wD:20.24,(3.33,3.85,;2,4.62,;.67,3.85,;-.67,4.62,;-2,3.85,;-2,2.31,;-3.33,1.54,;-4.67,2.31,;-6,1.54,;-6,,;-7.34,2.31,;-8.67,1.54,;-7.34,3.85,;-.67,1.54,;.67,2.31,;2,1.54,;2,,;3.33,-.77,;4.67,,;6,-.77,;6,-2.31,;4.67,-3.08,;3.33,-2.31,;7.34,-3.08,;8.67,-2.31,;7.34,-4.62,;8.67,-3.85,)| | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626319
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626361
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES OC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626358
(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)Show SMILES ONC(=O)C(=C)CNc1cc(-c2ccc(OC(F)(F)F)cc2)c2ncsc2c1C#N | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626360
(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626352
(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1CO)-c1ccc(OC(F)(F)F)cc1 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626365
(2-[[[7-cyano-4-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES ONC(=O)C(=C)CNc1cc(-c2ccc(cc2)S(F)(F)(F)(F)F)c2ncsc2c1C#N | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626318
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626324
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)NO)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626329
(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(=O)NO)c(CO)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626333
(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)Show SMILES OC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM50547124
(CHEMBL242708 | NCI-0001009) | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| Article
PubMed
| n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description
Inhibition of CPM binding to N-terminal His6-tagged human TEAD3 (216 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p... |
Citation and Details
Article DOI: 10.1021/acs.jmedchem.0c01275
BindingDB Entry DOI: 10.7270/Q2QN6BC1 |
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626363
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626364
(2-[[[4-cyano-7-(5-isopropylthiazol- 2-yl)-2,3-dih...)Show SMILES CC(C)c1cnc(s1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626318
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 2.88E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626331
(US11787775, Compound 16-C)Show SMILES C[C@@H](c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12)C(F)(F)F |r| | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626319
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)c(C#N)c2CCOc12 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626352
(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1CO)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626330
(2-[[[4-cyano-7-[4- (trifluoromethyl)phenyl]-2,3- ...)Show SMILES OC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)C(F)(F)F | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626335
(2-[[[4-(4-isopropylphenyl)-6,7- dihydrofuro[3,2-d...)Show SMILES CC(C)c1ccc(cc1)-c1nc(NCC(=C)C(O)=O)nc2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626336
(2-[[[4-fluoro-7-(4-isopropylphenyl)- 2,3-dihydrob...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(F)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626363
(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)Show SMILES NC(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(cc1)S(F)(F)(F)(F)F | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626342
(2-[[[4-cyano-7-(2-fluoro-4- isopropyl-phenyl)-2,3...)Show SMILES CC(C)c1ccc(c(F)c1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626332
(US11787775, Compound 16-D)Show SMILES C[C@H](c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12)C(F)(F)F |r| | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 6.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626334
(2-[[[4-cyano-7-[4-(1,1- difluoroethyl)phenyl]-2,3...)Show SMILES CC(F)(F)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 6.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626316
(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(O)=O)cc2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 8.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5/Isoform 5 of Transcriptional coactivator [50-100]
(Homo sapiens-Homo sapiens (Human)) | BDBM626359
(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)Show SMILES CN(O)C(=O)C(=C)CNc1cc(c2OCCc2c1C#N)-c1ccc(OC(F)(F)F)cc1 | PDB
UniProtKB/SwissProt
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 8.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626319
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626328
(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)Show SMILES CC(C)c1ccc(cc1)-c1cc(NCC(=C)C(N)=O)c(CO)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Transcriptional enhancer factor TEF-5
(Homo sapiens) | BDBM626322
(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)Show SMILES CC(C)c1ccc(cc1)-c1cc(N(C)CC(=C)C(O)=O)c(C#N)c2CCOc12 | PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
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