Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Inosine-adenosine-guanosine-nucleoside hydrolase (Trypanosoma brucei brucei) | BDBM50187701 (CHEMBL3827395) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Medical University of Lodz Curated by ChEMBL | Assay Description Inhibition of Trypanosoma brucei brucei inosine-adenosine-guanosine nucleoside hydrolase expressed in Escherichia coli | Eur J Med Chem 118: 121-42 (2016) Article DOI: 10.1016/j.ejmech.2016.04.034 BindingDB Entry DOI: 10.7270/Q2ZP482X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inosine-adenosine-guanosine-nucleoside hydrolase (Trypanosoma brucei brucei) | BDBM50187703 (CHEMBL3827853) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Medical University of Lodz Curated by ChEMBL | Assay Description Inhibition of Trypanosoma brucei brucei inosine-adenosine-guanosine nucleoside hydrolase expressed in Escherichia coli | Eur J Med Chem 118: 121-42 (2016) Article DOI: 10.1016/j.ejmech.2016.04.034 BindingDB Entry DOI: 10.7270/Q2ZP482X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inosine-adenosine-guanosine-nucleoside hydrolase (Trypanosoma brucei brucei) | BDBM50187702 (CHEMBL3828258) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Medical University of Lodz Curated by ChEMBL | Assay Description Inhibition of Trypanosoma brucei brucei inosine-adenosine-guanosine nucleoside hydrolase expressed in Escherichia coli | Eur J Med Chem 118: 121-42 (2016) Article DOI: 10.1016/j.ejmech.2016.04.034 BindingDB Entry DOI: 10.7270/Q2ZP482X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Inosine-adenosine-guanosine-nucleoside hydrolase (Trypanosoma brucei brucei) | BDBM50187700 (CHEMBL3828042) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Medical University of Lodz Curated by ChEMBL | Assay Description Inhibition of Trypanosoma brucei brucei inosine-adenosine-guanosine nucleoside hydrolase expressed in Escherichia coli | Eur J Med Chem 118: 121-42 (2016) Article DOI: 10.1016/j.ejmech.2016.04.034 BindingDB Entry DOI: 10.7270/Q2ZP482X | |||||||||||
More data for this Ligand-Target Pair |