Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223477 (US9320734, 316) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 1.74E+3 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223486 (US9320734, 331) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223488 (US9320734, 332) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223487 (US9320734, 333) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223489 (US9320734, 360) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223490 (US9320734, 335) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 980 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223477 (US9320734, 316) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 3.13E+4 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223486 (US9320734, 331) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223488 (US9320734, 332) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 3.57E+3 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223489 (US9320734, 360) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
3-phosphoinositide-dependent protein kinase 1 [409-556] (Homo sapiens (Human)) | BDBM223490 (US9320734, 335) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | 1.45E+3 | n/a | n/a | n/a | n/a | n/a |
Board of Regents, The University of Texas System; Arizona Board of Regents on behalf of the University of Arizona US Patent | Assay Description KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T... | US Patent US9320734 (2016) BindingDB Entry DOI: 10.7270/Q2QF8RRM | |||||||||||
More data for this Ligand-Target Pair |