Found 286 hits Enz. Inhib. hit(s) with Target = 'Probable G-protein coupled receptor 142' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50395775
(CHEMBL2164857)Show SMILES CNc1cc(ccn1)-c1nnc(NC(=O)[C@H](Cc2ccccc2)NCc2cscn2)s1 |r| Show InChI InChI=1S/C21H21N7OS2/c1-22-18-10-15(7-8-23-18)20-27-28-21(31-20)26-19(29)17(9-14-5-3-2-4-6-14)24-11-16-12-30-13-25-16/h2-8,10,12-13,17,24H,9,11H2,1H3,(H,22,23)(H,26,28,29)/t17-/m0/s1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen Inc
Curated by ChEMBL
| Assay Description Partial agonist activity at mouse GPR142 expressed in HEK293 cells |
Bioorg Med Chem Lett 22: 6218-23 (2012)
Article DOI: 10.1016/j.bmcl.2012.08.015 BindingDB Entry DOI: 10.7270/Q2CN751R |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558172
(CHEMBL4750179)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(Cl)c4)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558167
(CHEMBL4798957)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(OC(F)(F)F)c4)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558171
(CHEMBL4790150)Show SMILES FC(F)(F)c1cccc(Nc2nnc3-c4cc(ccc4OCCn23)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558161
(CHEMBL4746135)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4cccc(Cl)c4F)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558165
(CHEMBL4761139)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4cccc(Cl)c4)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558195
(CHEMBL4800653)Show SMILES Fc1c(Cl)cccc1NC(=O)N1CCOc2ccc(cc2C1)-c1ccncc1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 59 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558200
(CHEMBL4785678)Show SMILES O=C(Nc1cccc(c1)-c1ccccc1)N1CCOc2ccc(cc2C1)-c1ccncc1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558168
(CHEMBL4755454)Show SMILES FC(F)(F)Oc1cccc(Nc2nnc3-c4cc(ccc4OCCn23)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558170
(CHEMBL4788072)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(c4)C(F)(F)F)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558169
(CHEMBL4752684)Show SMILES CCc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(c4)C(F)(F)F)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 74 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558164
(CHEMBL4751613)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4cccc(OC(F)(F)F)c4)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 78 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558199
(CHEMBL4763234)Show SMILES O=C(Nc1cccc(c1)C#N)N1CCOc2ccc(cc2C1)-c1ccncc1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558199
(CHEMBL4763234)Show SMILES O=C(Nc1cccc(c1)C#N)N1CCOc2ccc(cc2C1)-c1ccncc1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558163
(CHEMBL4743615)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4ccccc4OC(F)(F)F)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558206
(CHEMBL4760456) | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 92 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558162
(CHEMBL4759692)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4ccccc4Cl)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 102 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558174
(CHEMBL4787638)Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 108 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558177
(CHEMBL4783052)Show SMILES O=C(Nc1cccc(c1)C#N)N1CCOc2ccc(cc2C1)-n1ccnc1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558198
(CHEMBL4756319)Show SMILES FC(F)(F)c1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558193
(CHEMBL4753373)Show SMILES Fc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 132 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558173
(CHEMBL4755668)Show SMILES Clc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 138 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558173
(CHEMBL4755668)Show SMILES Clc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558197
(CHEMBL4756931)Show SMILES O=C(Nc1cccc(Oc2ccccc2)c1)N1CCOc2ccc(cc2C1)-c1ccncc1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 146 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558190
(CHEMBL4782723)Show SMILES Clc1ccc(NC(=O)N2CCNc3ccc(cc3C2)-c2ccncc2)cc1Cl | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 146 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558191
(CHEMBL4751751)Show SMILES FC(F)(F)c1cccc(CS(=O)(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 157 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558194
(CHEMBL4754434)Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1Cl | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 157 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558198
(CHEMBL4756319)Show SMILES FC(F)(F)c1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 158 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558190
(CHEMBL4782723)Show SMILES Clc1ccc(NC(=O)N2CCNc3ccc(cc3C2)-c2ccncc2)cc1Cl | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 158 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558195
(CHEMBL4800653)Show SMILES Fc1c(Cl)cccc1NC(=O)N1CCOc2ccc(cc2C1)-c1ccncc1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 163 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558174
(CHEMBL4787638)Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 164 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558178
(CHEMBL4750165)Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2OC)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 187 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558176
(CHEMBL4779679)Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccnc3ccccc23)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 216 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558201
(CHEMBL4792959)Show SMILES Fc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 224 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558202
(CHEMBL4750832)Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 249 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558202
(CHEMBL4750832)Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 305 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558200
(CHEMBL4785678)Show SMILES O=C(Nc1cccc(c1)-c1ccccc1)N1CCOc2ccc(cc2C1)-c1ccncc1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 343 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558182
(CHEMBL4782047)Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccnc(C)c2)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 374 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558179
(CHEMBL4790417)Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2C)c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 394 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558201
(CHEMBL4792959)Show SMILES Fc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 413 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558180
(CHEMBL4781458)Show SMILES Nc1cc(ccn1)-c1ccc2OCCN(Cc2c1)C(=O)Nc1cccc(c1)C#N | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 448 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558178
(CHEMBL4750165)Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2OC)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 486 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558206
(CHEMBL4760456) | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 517 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558187
(CHEMBL4743675)Show SMILES Clc1ccc(NC(=O)N2CCCc3ccc(cc3C2)-c2ccncc2)cc1Cl | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 590 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558166
(CHEMBL4744842)Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Cc4cccc(Cl)c4)nnc3-c2c1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 593 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558205
(CHEMBL4781462) | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 604 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558192
(CHEMBL4781022)Show SMILES FC(F)(F)c1cccc(CC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1 | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 611 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Mus musculus) | BDBM50558193
(CHEMBL4753373)Show SMILES Fc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl | KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 613 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558194
(CHEMBL4754434)Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1Cl | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 708 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |
Probable G-protein coupled receptor 142
(Homo sapiens (Human)) | BDBM50558207
(CHEMBL4779820) | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 793 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| Assay Description Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay |
Citation and Details
Article DOI: 10.1016/j.bmcl.2016.04.018 BindingDB Entry DOI: 10.7270/Q2HM5D44 |
More data for this Ligand-Target Pair | |