BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 286 hits Enz. Inhib. hit(s) with Target = 'Probable G-protein coupled receptor 142'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50395775
PNG
(CHEMBL2164857)
Show SMILES CNc1cc(ccn1)-c1nnc(NC(=O)[C@H](Cc2ccccc2)NCc2cscn2)s1 |r|
Show InChI InChI=1S/C21H21N7OS2/c1-22-18-10-15(7-8-23-18)20-27-28-21(31-20)26-19(29)17(9-14-5-3-2-4-6-14)24-11-16-12-30-13-25-16/h2-8,10,12-13,17,24H,9,11H2,1H3,(H,22,23)(H,26,28,29)/t17-/m0/s1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 15n/an/an/an/an/an/a



Amgen Inc

Curated by ChEMBL


Assay Description
Partial agonist activity at mouse GPR142 expressed in HEK293 cells


Bioorg Med Chem Lett 22: 6218-23 (2012)


Article DOI: 10.1016/j.bmcl.2012.08.015
BindingDB Entry DOI: 10.7270/Q2CN751R
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558172
PNG
(CHEMBL4750179)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(Cl)c4)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 37n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558167
PNG
(CHEMBL4798957)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(OC(F)(F)F)c4)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 45n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558171
PNG
(CHEMBL4790150)
Show SMILES FC(F)(F)c1cccc(Nc2nnc3-c4cc(ccc4OCCn23)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 48n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558161
PNG
(CHEMBL4746135)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4cccc(Cl)c4F)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 56n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558165
PNG
(CHEMBL4761139)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4cccc(Cl)c4)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 58n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558195
PNG
(CHEMBL4800653)
Show SMILES Fc1c(Cl)cccc1NC(=O)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 59n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558200
PNG
(CHEMBL4785678)
Show SMILES O=C(Nc1cccc(c1)-c1ccccc1)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 62n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558168
PNG
(CHEMBL4755454)
Show SMILES FC(F)(F)Oc1cccc(Nc2nnc3-c4cc(ccc4OCCn23)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 63n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558170
PNG
(CHEMBL4788072)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(c4)C(F)(F)F)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 63n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558169
PNG
(CHEMBL4752684)
Show SMILES CCc1cc(ccn1)-c1ccc2OCCn3c(Nc4cccc(c4)C(F)(F)F)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 74n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558164
PNG
(CHEMBL4751613)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4cccc(OC(F)(F)F)c4)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 78n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558199
PNG
(CHEMBL4763234)
Show SMILES O=C(Nc1cccc(c1)C#N)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 79n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558199
PNG
(CHEMBL4763234)
Show SMILES O=C(Nc1cccc(c1)C#N)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 80n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558163
PNG
(CHEMBL4743615)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4ccccc4OC(F)(F)F)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 89n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558206
PNG
(CHEMBL4760456)
Show SMILES COc1ccccc1NC(=O)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 92n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558162
PNG
(CHEMBL4759692)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Oc4ccccc4Cl)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 102n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558174
PNG
(CHEMBL4787638)
Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 108n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558177
PNG
(CHEMBL4783052)
Show SMILES O=C(Nc1cccc(c1)C#N)N1CCOc2ccc(cc2C1)-n1ccnc1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 110n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558198
PNG
(CHEMBL4756319)
Show SMILES FC(F)(F)c1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 110n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558193
PNG
(CHEMBL4753373)
Show SMILES Fc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 132n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558173
PNG
(CHEMBL4755668)
Show SMILES Clc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 138n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558173
PNG
(CHEMBL4755668)
Show SMILES Clc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 140n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558197
PNG
(CHEMBL4756931)
Show SMILES O=C(Nc1cccc(Oc2ccccc2)c1)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 146n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558190
PNG
(CHEMBL4782723)
Show SMILES Clc1ccc(NC(=O)N2CCNc3ccc(cc3C2)-c2ccncc2)cc1Cl
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 146n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558191
PNG
(CHEMBL4751751)
Show SMILES FC(F)(F)c1cccc(CS(=O)(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 157n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558194
PNG
(CHEMBL4754434)
Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1Cl
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 157n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558198
PNG
(CHEMBL4756319)
Show SMILES FC(F)(F)c1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 158n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558190
PNG
(CHEMBL4782723)
Show SMILES Clc1ccc(NC(=O)N2CCNc3ccc(cc3C2)-c2ccncc2)cc1Cl
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 158n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558195
PNG
(CHEMBL4800653)
Show SMILES Fc1c(Cl)cccc1NC(=O)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 163n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558174
PNG
(CHEMBL4787638)
Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 164n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558178
PNG
(CHEMBL4750165)
Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2OC)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 187n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558176
PNG
(CHEMBL4779679)
Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccnc3ccccc23)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 216n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558201
PNG
(CHEMBL4792959)
Show SMILES Fc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 224n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558202
PNG
(CHEMBL4750832)
Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 249n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558202
PNG
(CHEMBL4750832)
Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 305n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558200
PNG
(CHEMBL4785678)
Show SMILES O=C(Nc1cccc(c1)-c1ccccc1)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 343n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558182
PNG
(CHEMBL4782047)
Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccnc(C)c2)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 374n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558179
PNG
(CHEMBL4790417)
Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2C)c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 394n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558201
PNG
(CHEMBL4792959)
Show SMILES Fc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 413n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558180
PNG
(CHEMBL4781458)
Show SMILES Nc1cc(ccn1)-c1ccc2OCCN(Cc2c1)C(=O)Nc1cccc(c1)C#N
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 448n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558178
PNG
(CHEMBL4750165)
Show SMILES COc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2OC)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 486n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558206
PNG
(CHEMBL4760456)
Show SMILES COc1ccccc1NC(=O)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 517n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558187
PNG
(CHEMBL4743675)
Show SMILES Clc1ccc(NC(=O)N2CCCc3ccc(cc3C2)-c2ccncc2)cc1Cl
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 590n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558166
PNG
(CHEMBL4744842)
Show SMILES Cc1cc(ccn1)-c1ccc2OCCn3c(Cc4cccc(Cl)c4)nnc3-c2c1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 593n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558205
PNG
(CHEMBL4781462)
Show SMILES Fc1ccccc1NC(=O)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 604n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558192
PNG
(CHEMBL4781022)
Show SMILES FC(F)(F)c1cccc(CC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 611n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Mus musculus)
BDBM50558193
PNG
(CHEMBL4753373)
Show SMILES Fc1ccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)cc1Cl
KEGG

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 613n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at mouse GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558194
PNG
(CHEMBL4754434)
Show SMILES Clc1cccc(NC(=O)N2CCOc3ccc(cc3C2)-c2ccncc2)c1Cl
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 708n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Probable G-protein coupled receptor 142


(Homo sapiens (Human))
BDBM50558207
PNG
(CHEMBL4779820)
Show SMILES O=C(Nc1ccccc1)N1CCOc2ccc(cc2C1)-c1ccncc1
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 793n/an/an/an/an/an/a


TBA

Assay Description
Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2016.04.018
BindingDB Entry DOI: 10.7270/Q2HM5D44
More data for this
Ligand-Target Pair
Displayed 1 to 50 (of 286 total )  |  Next  |  Last  >>
Jump to: