Compile Data Set for Download or QSAR

Found 122 hits Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 5'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50602136 (CHEMBL5183139) Show SMILES COc1ccc(\C=N\NC(=O)C2CC2c2ccccc2)cc1OC Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details Article DOI: 10.1016/j.bmc.2022.117084 BindingDB Entry DOI: 10.7270/Q2XW4PWD
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50602137 (CHEMBL5196998) Show SMILES COc1ccc(\C=N\NC(=O)Cc2cccc3ccccc23)cc1OC Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid PDB UniChem	Article PubMed	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details Article DOI: 10.1016/j.bmc.2022.117084 BindingDB Entry DOI: 10.7270/Q2XW4PWD
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50044849 (CHEMBL3311308) Show SMILES COc1ccc(cc1)S(=O)(=O)Nc1c(C)cc(C)cc1C Show InChI InChI=1S/C16H19NO3S/c1-11-9-12(2)16(13(3)10-11)17-21(18,19)15-7-5-14(20-4)6-8-15/h5-10,17H,1-4H3	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	<3.98E+4	n/a	n/a	n/a	n/a	n/a	n/a
GlaxoSmithKline Curated by ChEMBL					Assay Description Blocking of human TRPM5 expressed in HEK293 cells by FLIPR membrane potential/summary (Abse5) assay				Bioorg Med Chem Lett 24: 3100-3 (2014) Article DOI: 10.1016/j.bmcl.2014.05.012 BindingDB Entry DOI: 10.7270/Q2CC1292
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50044849 (CHEMBL3311308) Show SMILES COc1ccc(cc1)S(=O)(=O)Nc1c(C)cc(C)cc1C Show InChI InChI=1S/C16H19NO3S/c1-11-9-12(2)16(13(3)10-11)17-21(18,19)15-7-5-14(20-4)6-8-15/h5-10,17H,1-4H3	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	<5.01E+4	n/a	n/a	n/a	n/a
GlaxoSmithKline Curated by ChEMBL					Assay Description Induction of human TRPM5 opening expressed in HEK293 cells by FLIPR membrane potential/summary (Abse5) assay				Bioorg Med Chem Lett 24: 3100-3 (2014) Article DOI: 10.1016/j.bmcl.2014.05.012 BindingDB Entry DOI: 10.7270/Q2CC1292
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571574 (CHEMBL4873144) Show SMILES Cn1c(Cl)cnc1CNc1ccc(Cl)cc1F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	4.68E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571570 (CHEMBL4876211) Show SMILES Cn1c(Cl)cnc1CNc1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	331	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571575 (CHEMBL4858947) Show SMILES COc1ccc(cc1OC)N(C)Cc1ncc(Cl)n1C Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571576 (CHEMBL4877096) Show SMILES Cn1c(Cl)cnc1CN1CCc2ccccc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	2.29E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571577 (CHEMBL4853398) Show SMILES Cn1ccnc1CNc1ccc(Cl)cc1OCCC(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	2.51E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571578 (CHEMBL4870747) Show SMILES Cn1c(Cl)cnc1CN1CC(CO)Cc2cccc(F)c12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	5.01E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571579 (CHEMBL4873490) Show SMILES CCN(Cc1ncc(Cl)n1C)c1ccc(Br)cc1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	5.13E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571580 (CHEMBL1440011) Show SMILES Cn1c(CNc2ccc(Cl)cc2)nc2ccccc12 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571581 (CHEMBL4855094) Show SMILES Cn1c(Cl)cnc1CNc1ccc2oncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	3.02E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571582 (CHEMBL4876435) Show SMILES Cn1c(Cl)cnc1CNc1ccc2[nH]ncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	6.03E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571583 (CHEMBL4852732) Show SMILES Cn1c(Cl)cnc1CNc1ccc2n(C)ncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	5.25E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571584 (CHEMBL4868164) Show SMILES Cn1c(Cl)cnc1CNc1ccc2scnc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.35E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571585 (CHEMBL4847994) Show SMILES Cn1c(Cl)cnc1CNc1ccc2ocnc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.62E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571586 (CHEMBL4846618) Show SMILES Cn1c(Cl)cnc1CNc1ccc2[nH]cnc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571587 (CHEMBL4858831) Show SMILES Cn1c(Cl)cnc1CNc1ccc2n(C)nnc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571588 (CHEMBL4847928) Show SMILES Clc1cnc(CNc2ccc3sncc3c2)[nH]1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571589 (CHEMBL4849590) Show SMILES Cn1c(CNc2ccc3sncc3c2)nc(Cl)c1Cl Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571590 (CHEMBL4851802) Show SMILES Cn1ccnc1CNc1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	5.13E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571591 (CHEMBL4859679) Show SMILES Cn1c(Cl)ccc1CNc1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571592 (CHEMBL4855887) Show SMILES Cn1c(Br)cnc1CNc1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	457	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571593 (CHEMBL4877090) Show SMILES Clc1snnc1CNc1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	5.25E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571594 (CHEMBL4850328) Show SMILES Cc1nnc(CNc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	1.91E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571595 (CHEMBL4876532) Show SMILES Cn1nc(CNc2ccc3sncc3c2)cc1C(F)(F)F Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571596 (CHEMBL4855627) Show SMILES N#Cc1ccc(CNc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571571 (CHEMBL4849726) Show SMILES Clc1cnc(CNc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	89	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571597 (CHEMBL4871574) Show SMILES Clc1ccc(CNc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571598 (CHEMBL4874619) Show SMILES FC(F)(F)c1cnc(CNc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	490	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571599 (CHEMBL4866780) Show SMILES Cc1cnc(CNc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	575	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571600 (CHEMBL4849306) Show SMILES CC(C)c1cnc(CNc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571601 (CHEMBL4867233) Show SMILES Cc1csc(CNc2ccc3sncc3c2)n1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571602 (CHEMBL4853883) Show SMILES Cc1nc(CNc2ccc3sncc3c2)sc1C Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571603 (CHEMBL4857099) Show SMILES C(Nc1ccc2sncc2c1)c1nccs1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	4.68E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571604 (CHEMBL4872851) Show SMILES C(Nc1ccc2sncc2c1)c1nc2ccccc2s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571605 (CHEMBL4869736) Show SMILES CN(Cc1ncc(Cl)n1C)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	158	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571606 (CHEMBL4863555) Show SMILES CN(Cc1ncc(Cl)s1)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	447	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571607 (CHEMBL4863223) Show SMILES Cn1c(Cl)cnc1CN(CC1CC1)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	158	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571608 (CHEMBL4873210) Show SMILES CC(C)N(Cc1ncc(Cl)n1C)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	5.13E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571609 (CHEMBL4856537) Show SMILES Cn1c(Cl)cnc1CN(CC1CCCCC1)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571610 (CHEMBL4865623) Show SMILES Cn1c(Cl)cnc1CN(Cc1ccccc1)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571611 (CHEMBL4849797) Show SMILES CCN(Cc1ncc(Cl)n1C)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	468	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571612 (CHEMBL4875178) Show SMILES CC(=O)N(Cc1ncc(Cl)n1C)c1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571613 (CHEMBL4869125) Show SMILES Clc1cnc(s1)C(=O)Nc1ccc2sncc2c1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571614 (CHEMBL4861541) Show SMILES CC(Nc1ccc2sncc2c1)c1ncc(Cl)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	7.59E+3	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571615 (CHEMBL4850518) Show SMILES CC(C)(Nc1ccc2sncc2c1)c1ncc(Cl)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	<3.16E+4	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571616 (CHEMBL4867011) Show SMILES Clc1cnc(COc2ccc3sncc3c2)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	832	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 5 (Homo sapiens (Human))	BDBM50571617 (CHEMBL4860824) Show SMILES Cc1cc2sncc2cc1NCc1ncc(Cl)s1 Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	39	n/a	n/a	n/a	n/a
TBA					Assay Description Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assay				Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00065 BindingDB Entry DOI: 10.7270/Q2J106ZZ
					More data for this Ligand-Target Pair

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