Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cardiac ryanodine receptor 2 (Canis familiaris) | BDBM50044994 (2,6,9,11,13,14-hexahydroxy-11-isopropyl-3,7,10-tri...) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Binding affinity towards ryanodine receptor in canine ventrical preparation | J Med Chem 39: 2339-46 (1996) Article DOI: 10.1021/jm950712d BindingDB Entry DOI: 10.7270/Q2T15490 | |||||||||||
More data for this Ligand-Target Pair |