Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442747 (CHEMBL2443009) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442752 (CHEMBL2443004) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442750 (CHEMBL2443006) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442751 (CHEMBL2443005) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442746 (CHEMBL2443010) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442748 (CHEMBL2443008) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442749 (CHEMBL2443007) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442754 (CHEMBL2443002) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442756 (CHEMBL2443000) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442755 (CHEMBL2443001) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (Sus scrofa) | BDBM50442753 (CHEMBL2443003) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Friedrich-Alexander University Curated by ChEMBL | Assay Description Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortex | Bioorg Med Chem Lett 23: 6079-82 (2013) Article DOI: 10.1016/j.bmcl.2013.09.026 BindingDB Entry DOI: 10.7270/Q2028T08 | |||||||||||
More data for this Ligand-Target Pair |