Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Chemokine receptor (Oryctolagus cuniculus) | BDBM50399208 (CHEMBL2180528) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Company Curated by ChEMBL | Assay Description Displacement of [125I]MIP-1alpha from CCR1 in rabbit PBMCs incubated for 60 mins | J Med Chem 55: 9643-53 (2012) Article DOI: 10.1021/jm300896d BindingDB Entry DOI: 10.7270/Q2ST7R0S | |||||||||||
More data for this Ligand-Target Pair |