Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501358 (CHEMBL3947604) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469157 (CHEMBL4284736) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501352 (CHEMBL3922978) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469159 (CHEMBL4283840) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501354 (CHEMBL3934222) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469154 (CHEMBL4283678) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469165 (CHEMBL4291540) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469162 (CHEMBL4282733) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469170 (CHEMBL4291025) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 42 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501357 (CHEMBL3957297) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469166 (CHEMBL4294422) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469169 (CHEMBL4292925) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 72 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469164 (CHEMBL4287199) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 98 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469160 (CHEMBL4280386) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 104 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469167 (CHEMBL4279276) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 105 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469161 (CHEMBL4290610) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 107 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501351 (CHEMBL3924425) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469163 (CHEMBL4282334) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 175 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50480585 (CHEMBL555725) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Inhibition of Escherichia coli signal peptidase | Bioorg Med Chem Lett 19: 3787-90 (2009) Article DOI: 10.1016/j.bmcl.2009.04.034 BindingDB Entry DOI: 10.7270/Q2B27Z2J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469168 (CHEMBL4281328) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 225 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469156 (CHEMBL4291944) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 227 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501353 (CHEMBL3895001) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469158 (CHEMBL4280228) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 495 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501356 (CHEMBL2306366) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50469155 (CHEMBL4288133) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi... | Eur J Med Chem 157: 1346-1360 (2018) Article DOI: 10.1016/j.ejmech.2018.08.086 BindingDB Entry DOI: 10.7270/Q2H70JH1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501356 (CHEMBL2306366) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50480486 (CHEMBL539137) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.34E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Katholieke Universiteit Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type I signal peptidase lepB | Bioorg Med Chem Lett 19: 2880-3 (2009) Article DOI: 10.1016/j.bmcl.2009.03.064 BindingDB Entry DOI: 10.7270/Q2V40Z0B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50480486 (CHEMBL539137) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.34E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Katholieke Universiteit Leuven Curated by ChEMBL | Assay Description Inhibition of Escherichia coli type I signal peptidase lepB | Bioorg Med Chem Lett 19: 2880-3 (2009) Article DOI: 10.1016/j.bmcl.2009.03.064 BindingDB Entry DOI: 10.7270/Q2V40Z0B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50501355 (CHEMBL3952118) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Uppsala University Curated by ChEMBL | Assay Description Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra... | Bioorg Med Chem 25: 897-911 (2017) Article DOI: 10.1016/j.bmc.2016.12.003 BindingDB Entry DOI: 10.7270/Q20P1321 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50441139 (ARYLOMYCIN C16) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 979 | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Curated by ChEMBL | Assay Description Binding affinity to full length His-tagged Escherichia coli MG1665 SPase 1 expressed in Escherichia coli BL21 (DE3) | Bioorg Med Chem Lett 24: 413-8 (2014) Article DOI: 10.1016/j.bmcl.2013.12.059 BindingDB Entry DOI: 10.7270/Q29K4F5D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Signal peptidase I (Escherichia coli (strain K12)) | BDBM50441139 (ARYLOMYCIN C16) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 39 | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Curated by ChEMBL | Assay Description Binding affinity to full length His-tagged Escherichia coli PAS0232 SPase 1 P84S mutant expressed in Escherichia coli BL21 (DE3) | Bioorg Med Chem Lett 24: 413-8 (2014) Article DOI: 10.1016/j.bmcl.2013.12.059 BindingDB Entry DOI: 10.7270/Q29K4F5D | |||||||||||
More data for this Ligand-Target Pair |