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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Telomerase reverse transcriptase' AND taxid = 10116   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Telomerase reverse transcriptase


(Rattus norvegicus)		BDBM50446425
PNG
(CHEMBL3109741)
Show SMILES FC(F)(F)c1cccc(c1)-n1sccc1=O
Show InChI InChI=1S/C10H6F3NOS/c11-10(12,13)7-2-1-3-8(6-7)14-9(15)4-5-16-14/h1-6H
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CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 1.00E+3n/an/an/an/an/an/a



University of North Carolina at Chapel Hill

Curated by ChEMBL


Assay Description
Inhibition of rat telomerase by TRAP assay

J Med Chem 57: 521-38 (2014)


Article DOI: 10.1021/jm400528t
BindingDB Entry DOI: 10.7270/Q2T43VKJ
More data for this
Ligand-Target Pair