Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120757 (US8703761, 1-29) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120755 (US8703761, 1-8) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120756 (US8703761, 1-28) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120759 (US8703761, 8-1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 54.5 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120753 (US8703761, 1-1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 60.5 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120758 (US8703761, 6-14) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 197 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120763 (US8703761, 14-4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 225 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120760 (US8703761, 8-2) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 240 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120754 (US8703761, 1-6) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 241 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120767 (US8703761, 6-1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 910 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120761 (US8703761, 12-3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.18E+3 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120765 (US8703761, 14-24) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.75E+3 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120762 (US8703761, 12-4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.08E+3 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120764 (US8703761, 14-3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Diacylglycerol O-acyltransferase 1 [89-488] (Homo sapiens (Human)) | BDBM120766 (US8703761, 14-28) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.13E+3 | n/a | n/a | n/a | n/a | 7.5 | 4 |
Novartis AG US Patent | Assay Description The enzyme preparation used in this assay is a membrane preparation from Sf9 cells overexpressing human (His)6DGAT1. During all steps samples were ch... | US Patent US8703761 (2014) BindingDB Entry DOI: 10.7270/Q2057DM1 | |||||||||||
More data for this Ligand-Target Pair |