Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dual specificity mitogen-activated protein kinase kinase 4 (Mus musculus) | BDBM50396483 (PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | 8.20 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assay | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112963 BindingDB Entry DOI: 10.7270/Q2MW2MXG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity mitogen-activated protein kinase kinase 4 (Mus musculus) | BDBM50568580 (CHEMBL4857316) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assay | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112963 BindingDB Entry DOI: 10.7270/Q2MW2MXG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity mitogen-activated protein kinase kinase 4 (Mus musculus) | BDBM50568579 (CHEMBL4848804) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 0.850 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assay | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112963 BindingDB Entry DOI: 10.7270/Q2MW2MXG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity mitogen-activated protein kinase kinase 4 (Mus musculus) | BDBM50568578 (CHEMBL4868537) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assay | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112963 BindingDB Entry DOI: 10.7270/Q2MW2MXG | |||||||||||
More data for this Ligand-Target Pair |