Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 4 (Homo sapiens (Human)) | BDBM50049744 (CHEMBL438548 | NPY-analogs | [Cys-Trp-Arg-Nva-Arg-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 570 | n/a | n/a | n/a | n/a |
University of Cincinnati Curated by ChEMBL | Assay Description Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesis | J Med Chem 49: 2661-5 (2006) Article DOI: 10.1021/jm050907d BindingDB Entry DOI: 10.7270/Q2XS5TZ9 | |||||||||||
More data for this Ligand-Target Pair |