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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50140900   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Mu-type opioid receptor


(GUINEA PIG)		BDBM50140900
PNG
(6-(2,4-dichlorophenyl)-19-methyl-(2R,10R)-11-oxa-8...)
Show SMILES CN1CC[C@@]23[C@H]4Oc5c2c(CC1[C@@H]3Cc1cc(cnc41)-c1ccc(Cl)cc1Cl)ccc5O |TLB:28:9:12:1.3.2|
Show InChI InChI=1S/C26H22Cl2N2O2/c1-30-7-6-26-18-9-14-8-15(17-4-3-16(27)11-19(17)28)12-29-23(14)25(26)32-24-21(31)5-2-13(22(24)26)10-20(18)30/h2-5,8,11-12,18,20,25,31H,6-7,9-10H2,1H3/t18-,20?,25-,26-/m0/s1
PDB

UniProtKB/SwissProt

B.MOAD
GoogleScholar
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PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a 225n/an/an/an/a



Southern Research Institute

Curated by ChEMBL


Assay Description
Agonistic activity towards Opioid receptor mu 1 was determined in [35S]GTP-gamma-S, binding assay in guinea pig caudate; g = not active as an agonist

J Med Chem 47: 1400-12 (2004)


Article DOI: 10.1021/jm030311v
BindingDB Entry DOI: 10.7270/Q2639QGW
More data for this
Ligand-Target Pair