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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50152811   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM50152811
PNG
(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Show SMILES NCCNCc1ccccc1N1CCN(CC1)C(=O)[C@@H](Cc1ccc(Cl)cc1)NC(=O)[C@H]1Cc2ccccc2CN1
Show InChI InChI=1S/C32H39ClN6O2/c33-27-11-9-23(10-12-27)19-29(37-31(40)28-20-24-5-1-2-6-25(24)22-36-28)32(41)39-17-15-38(16-18-39)30-8-4-3-7-26(30)21-35-14-13-34/h1-12,28-29,35-36H,13-22,34H2,(H,37,40)/t28-,29-/m1/s1
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Article
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n/an/an/an/a 91n/an/an/an/a



Neurocrine Biosciences, Inc.

Curated by ChEMBL


Assay Description
Effective concentration against cAMP release in CHO cells expressing human melanocortin-4 receptor

Bioorg Med Chem Lett 14: 4417-23 (2004)


Article DOI: 10.1016/j.bmcl.2004.06.059
BindingDB Entry DOI: 10.7270/Q2251HPH
More data for this
Ligand-Target Pair