Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM50213770![]() (3-(4-(2-(benzyl(6-chlorobenzo[d]thiazol-2-yl)amino...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.36E+3 | n/a | n/a | n/a | n/a |
Nagoya City University Curated by ChEMBL | Assay Description Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assay | Bioorg Med Chem Lett 17: 4351-7 (2007) Article DOI: 10.1016/j.bmcl.2007.05.017 BindingDB Entry DOI: 10.7270/Q2WM1D41 | |||||||||||
More data for this Ligand-Target Pair |