Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM50297886 (2-(4-(3-(3-(trifluoromethyl)phenoxy)propoxy)phenyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
Goethe-University Frankfurt Curated by ChEMBL | Assay Description Agonist activity at human PPARalpha expressed in african green monkey COS7 cells by Gal4 transactivation assay | Bioorg Med Chem Lett 19: 4421-6 (2009) Article DOI: 10.1016/j.bmcl.2009.05.057 BindingDB Entry DOI: 10.7270/Q2G160W7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM50297886 (2-(4-(3-(3-(trifluoromethyl)phenoxy)propoxy)phenyl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.60E+3 | n/a | n/a | n/a | n/a |
Goethe-University Frankfurt Curated by ChEMBL | Assay Description Agonist activity at human PPARgamma expressed in african green monkey COS7 cells by Gal4 transactivation assay | Bioorg Med Chem Lett 19: 4421-6 (2009) Article DOI: 10.1016/j.bmcl.2009.05.057 BindingDB Entry DOI: 10.7270/Q2G160W7 | |||||||||||
More data for this Ligand-Target Pair |