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Compile Data Set for Download or QSAR

Found 1 hit of ec50 for monomerid = 50414690   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
5-hydroxytryptamine receptor 4


(Homo sapiens (Human))		BDBM50414690
PNG
(CHEMBL560876)
Show SMILES [H][C@@]12CC[C@]([H])(CC(C1)NC(=O)c1cc3ccccc3n(C(C)C)c1=O)N2CCCCCCCCO |r|
Show InChI InChI=1S/C28H41N3O3/c1-20(2)31-26-12-8-7-11-21(26)17-25(28(31)34)27(33)29-22-18-23-13-14-24(19-22)30(23)15-9-5-3-4-6-10-16-32/h7-8,11-12,17,20,22-24,32H,3-6,9-10,13-16,18-19H2,1-2H3,(H,29,33)/t23-,24-/m1/s1
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PC sid
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Similars
Article
PubMed
n/an/an/an/a 15.8n/an/an/an/a



Theravance, Inc.

Curated by ChEMBL


Assay Description
Agonist activity at human 5HT4C receptor expressed in HEK293 cells assessed as acumulation of cAMP by flash plate adenylyl cyclase activation assay

J Med Chem 52: 5330-43 (2009)


Article DOI: 10.1021/jm900881j
BindingDB Entry DOI: 10.7270/Q2CF9RBH
More data for this
Ligand-Target Pair