Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
L-lactate dehydrogenase B chain (Homo sapiens (Human)) | BDBM50420178 (GUANIDINE) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.33E+8 | n/a | n/a | n/a | n/a |
Universit£ Catholique de Louvain (UCLouvain) Curated by ChEMBL | Assay Description Binding affinity full length human N-terminal His6-tagged LDH-H I8A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt... | J Med Chem 63: 4628-4643 (2020) Article DOI: 10.1021/acs.jmedchem.9b01955 BindingDB Entry DOI: 10.7270/Q2TB1BCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
L-lactate dehydrogenase B chain (Homo sapiens (Human)) | BDBM50420178 (GUANIDINE) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6.24E+8 | n/a | n/a | n/a | n/a |
Universit£ Catholique de Louvain (UCLouvain) Curated by ChEMBL | Assay Description Binding affinity full length human N-terminal His6-tagged LDH-H L3A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt... | J Med Chem 63: 4628-4643 (2020) Article DOI: 10.1021/acs.jmedchem.9b01955 BindingDB Entry DOI: 10.7270/Q2TB1BCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
L-lactate dehydrogenase B chain (Homo sapiens (Human)) | BDBM50420178 (GUANIDINE) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.54E+8 | n/a | n/a | n/a | n/a |
Universit£ Catholique de Louvain (UCLouvain) Curated by ChEMBL | Assay Description Binding affinity full length human N-terminal His6-tagged LDH-H K6A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt... | J Med Chem 63: 4628-4643 (2020) Article DOI: 10.1021/acs.jmedchem.9b01955 BindingDB Entry DOI: 10.7270/Q2TB1BCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
L-lactate dehydrogenase B chain (Homo sapiens (Human)) | BDBM50420178 (GUANIDINE) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.78E+8 | n/a | n/a | n/a | n/a |
Universit£ Catholique de Louvain (UCLouvain) Curated by ChEMBL | Assay Description Binding affinity full length human N-terminal His6-tagged LDH-H T2A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt... | J Med Chem 63: 4628-4643 (2020) Article DOI: 10.1021/acs.jmedchem.9b01955 BindingDB Entry DOI: 10.7270/Q2TB1BCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
L-lactate dehydrogenase B chain (Homo sapiens (Human)) | BDBM50420178 (GUANIDINE) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.91E+8 | n/a | n/a | n/a | n/a |
Universit£ Catholique de Louvain (UCLouvain) Curated by ChEMBL | Assay Description Binding affinity full length human N-terminal His6-tagged LDH-H K4A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt... | J Med Chem 63: 4628-4643 (2020) Article DOI: 10.1021/acs.jmedchem.9b01955 BindingDB Entry DOI: 10.7270/Q2TB1BCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
L-lactate dehydrogenase B chain (Homo sapiens (Human)) | BDBM50420178 (GUANIDINE) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.01E+9 | n/a | n/a | n/a | n/a |
Universit£ Catholique de Louvain (UCLouvain) Curated by ChEMBL | Assay Description Binding affinity full length human N-terminal His6-tagged LDH-H E5A mutant expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disrupt... | J Med Chem 63: 4628-4643 (2020) Article DOI: 10.1021/acs.jmedchem.9b01955 BindingDB Entry DOI: 10.7270/Q2TB1BCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
L-lactate dehydrogenase B chain (Homo sapiens (Human)) | BDBM50420178 (GUANIDINE) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.11E+9 | n/a | n/a | n/a | n/a |
Universit£ Catholique de Louvain (UCLouvain) Curated by ChEMBL | Assay Description Binding affinity to full length human N-terminal His6-tagged LDH-H expressed in Escherichia coli Rosetta (DE3) assessed as tetrameric disruption by n... | J Med Chem 63: 4628-4643 (2020) Article DOI: 10.1021/acs.jmedchem.9b01955 BindingDB Entry DOI: 10.7270/Q2TB1BCZ | |||||||||||
More data for this Ligand-Target Pair |