Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463353 (CHEMBL4248974) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463352 (CHEMBL4238053) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463354 (CHEMBL4246320) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463359 (CHEMBL4243509) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463351 (CHEMBL4240212) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463353 (CHEMBL4248974) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Activation of p53 in human MCF7 cell lysates assessed as increase in total p53 protein level by Western blot analysis | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463358 (CHEMBL4244338) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 65 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463356 (CHEMBL4240141) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 74 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463355 (CHEMBL4240977) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 152 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463357 (CHEMBL4243377) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 158 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cellular tumor antigen p53 (Homo sapiens (Human)) | BDBM50463350 (CHEMBL4243580) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Induction of p53 transcriptional activity (unknown origin) expressed in HEK293 cells coexpressing TK-driven Rluc after 20 to 22 hrs by luciferase rep... | Bioorg Med Chem 26: 4441-4451 (2018) Article DOI: 10.1016/j.bmc.2018.07.042 BindingDB Entry DOI: 10.7270/Q2CN76JW | |||||||||||
More data for this Ligand-Target Pair |