Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
14-3-3 protein zeta/delta (Homo sapiens) | BDBM50540834 (CHEMBL4640360) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+5 | n/a | n/a | n/a | n/a |
University of Groningen Curated by ChEMBL | Assay Description Binding affinity to 14-3-3 zeta (unknown origin) assessed as 14-3-3 zeta-synaptopodin interaction by fluorescence polarization assay | ACS Med Chem Lett 11: 1041-1046 (2020) Article DOI: 10.1021/acsmedchemlett.9b00541 BindingDB Entry DOI: 10.7270/Q24B34V9 | |||||||||||
More data for this Ligand-Target Pair |