Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3/cAMP-dependent protein kinase (Homo sapiens (Human)-Oryctolagus cuniculus (Rabbit...) | BDBM50169892 (3-{4-[4-(3-Chloro-phenylamino)-[1,3,5]triazin-2-yl...) | PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of Cyclin-dependent kinase 1-cyclin B | J Med Chem 48: 4535-46 (2005) Article DOI: 10.1021/jm040214h BindingDB Entry DOI: 10.7270/Q2833RK0 | |||||||||||
More data for this Ligand-Target Pair |