Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095321 (2-Methoxy-5-(3,4,5-trimethoxy-benzyloxy)-benzaldeh...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Effect on tubulin binding and the concentration required to cause 50% decrease in tubulin assembly at 350 nm. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50135466 (CHEMBL3752997) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arkansas for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by spectrophotometric analysis | Medchemcomm 6: 1535-1543 (2016) BindingDB Entry DOI: 10.7270/Q2H41T8J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095321 (2-Methoxy-5-(3,4,5-trimethoxy-benzyloxy)-benzaldeh...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Concentration required to cause 50% decrease in the binding of [3H]colchicine from purified porcine tubulin. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095317 (2-Methoxy-5-(3,4,5-trimethoxy-phenoxymethyl)-pheno...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Effect on tubulin binding and the concentration required to cause 50% decrease in tubulin assembly at 350 nm. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50135464 (CHEMBL3753885) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.35E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arkansas for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by spectrophotometric analysis | Medchemcomm 6: 1535-1543 (2016) BindingDB Entry DOI: 10.7270/Q2H41T8J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095326 (2-Methoxy-5-(3,4,5-trimethoxy-phenoxy)-phenol | CH...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.63E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Effect on tubulin binding and the concentration required to cause 50% decrease in tubulin assembly at 350 nm. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50135465 (CHEMBL3753880) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.85E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Arkansas for Medical Sciences Curated by ChEMBL | Assay Description Inhibition of porcine brain tubulin polymerization by spectrophotometric analysis | Medchemcomm 6: 1535-1543 (2016) BindingDB Entry DOI: 10.7270/Q2H41T8J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095320 (2-Methoxy-5-(3,4,5-trimethoxy-benzyloxy)-phenol | ...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Effect on tubulin binding and the concentration required to cause 50% decrease in tubulin assembly at 350 nm. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095326 (2-Methoxy-5-(3,4,5-trimethoxy-phenoxy)-phenol | CH...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Concentration required to cause 50% decrease in the binding of [3H]colchicine from purified porcine tubulin. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095317 (2-Methoxy-5-(3,4,5-trimethoxy-phenoxymethyl)-pheno...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Concentration required to cause 50% decrease in the binding of [3H]colchicine from purified porcine tubulin. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50134459 (2-(3-Hydroxy-4-methoxy-phenyl)-6,7,8-trimethoxy-ch...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiff University Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]colchicine to porcine tubulin | Bioorg Med Chem Lett 13: 3759-63 (2003) BindingDB Entry DOI: 10.7270/Q2G73D48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50134450 (2-[1-(3-Hydroxy-4-methoxy-phenyl)-meth-(Z)-ylidene...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Cardiff University Curated by ChEMBL | Assay Description Ability to inhibit the binding of [3H]colchicine to porcine tubulin | Bioorg Med Chem Lett 13: 3759-63 (2003) BindingDB Entry DOI: 10.7270/Q2G73D48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095319 (2-Methoxy-5-(3,4,5-trimethoxy-phenylamino)-phenol ...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Effect on tubulin binding and the concentration required to cause 50% decrease in tubulin assembly at 350 nm. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095320 (2-Methoxy-5-(3,4,5-trimethoxy-benzyloxy)-phenol | ...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.26E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Concentration required to cause 50% decrease in the binding of [3H]colchicine from purified porcine tubulin. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tubulin alpha-1A/beta chain (Sus scrofa (Pig)) | BDBM50095319 (2-Methoxy-5-(3,4,5-trimethoxy-phenylamino)-phenol ...) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.98E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Manchester Curated by ChEMBL | Assay Description Concentration required to cause 50% decrease in the binding of [3H]colchicine from purified porcine tubulin. | Bioorg Med Chem Lett 11: 51-4 (2001) BindingDB Entry DOI: 10.7270/Q2C82CHT | |||||||||||
More data for this Ligand-Target Pair |