Compile Data Set for Download or QSAR

Found 4 hits of ic50 for monomerid = 429578   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Proteinase-activated receptor 2 (Homo sapiens (Human))	BDBM429578 (US10550089, Example 52 | US10995072, Example 52) Show SMILES Cc1coc2c(F)ccc(C(O)c3ncc[nH]3)c12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	970	n/a	n/a	n/a	n/a	n/a	n/a
Heptares Therapeutics Limited US Patent					Assay Description Inositol monophosphate (IP1) production were measured in 1321N1 cells stably expressing human PAR2 using an IP-One HTRF assay kit (Cisbio). 80 nl of ...				US Patent US10995072 (2021) BindingDB Entry DOI: 10.7270/Q2D79FJQ
					More data for this Ligand-Target Pair
Proteinase-activated receptor 2 (Homo sapiens (Human))	BDBM429578 (US10550089, Example 52 | US10995072, Example 52) Show SMILES Cc1coc2c(F)ccc(C(O)c3ncc[nH]3)c12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.63E+3	n/a	n/a	n/a	n/a	n/a	n/a
Heptares Therapeutics Limited US Patent					Assay Description Inositol monophosphate (IP1) production were measured in 1321N1 cells stably expressing human PAR2 using an IP-One HTRF assay kit (Cisbio). 80 nl of ...				US Patent US10550089 (2020) BindingDB Entry DOI: 10.7270/Q2SB484T
					More data for this Ligand-Target Pair
Proteinase-activated receptor 2 (Homo sapiens (Human))	BDBM429578 (US10550089, Example 52 | US10995072, Example 52) Show SMILES Cc1coc2c(F)ccc(C(O)c3ncc[nH]3)c12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	3.27E+3	n/a	n/a	n/a	n/a	n/a	n/a
Heptares Therapeutics Limited US Patent					Assay Description Calcium mobilization was measured using 1321N1 cells stably expressing human PAR2. Cells were seeded in 384-well plates at 4,000 cells per well in 20...				US Patent US10995072 (2021) BindingDB Entry DOI: 10.7270/Q2D79FJQ
					More data for this Ligand-Target Pair
Proteinase-activated receptor 2 (Homo sapiens (Human))	BDBM429578 (US10550089, Example 52 | US10995072, Example 52) Show SMILES Cc1coc2c(F)ccc(C(O)c3ncc[nH]3)c12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	5.42E+3	n/a	n/a	n/a	n/a	n/a	n/a
Heptares Therapeutics Limited US Patent					Assay Description Calcium mobilization was measured using 1321N1 cells stably expressing human PAR2. Cells were seeded in 384-well plates at 4,000 cells per well in 20...				US Patent US10550089 (2020) BindingDB Entry DOI: 10.7270/Q2SB484T
					More data for this Ligand-Target Pair