Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
PAS domain-containing serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM463458![]() (3-(4-Fluorophenyl)-2-(4-(4-methoxyphenyl)piperidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
BioEnergenix LLC US Patent | Assay Description Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D... | US Patent US10781185 (2020) BindingDB Entry DOI: 10.7270/Q2DR2ZKW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PAS domain-containing serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM463458![]() (3-(4-Fluorophenyl)-2-(4-(4-methoxyphenyl)piperidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
BioEnergenix LLC US Patent | Assay Description Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i... | US Patent US10781185 (2020) BindingDB Entry DOI: 10.7270/Q2DR2ZKW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PAS domain-containing serine/threonine-protein kinase (Homo sapiens (Human)) | BDBM463458![]() (3-(4-Fluorophenyl)-2-(4-(4-methoxyphenyl)piperidin...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description One assay for purified hPASK activity utilizes the Kinase-Glo Luminescent Kinase Assay (Promega), which quantifies the amount of ATP remaining in sol... | Citation and Details BindingDB Entry DOI: 10.7270/Q2D79FN2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
PAS domain-containing serine/threonine-protein kinase [879-1323] (Homo sapiens (Human)) | BDBM463458![]() (3-(4-Fluorophenyl)-2-(4-(4-methoxyphenyl)piperidin...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is... | Citation and Details BindingDB Entry DOI: 10.7270/Q2D79FN2 | |||||||||||
More data for this Ligand-Target Pair |