Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50154863![]() (CHEMBL3775256 | US10273244, Example 162 | US105841...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >100 | n/a | n/a | n/a | n/a | n/a | n/a |
Aptuit s.r.l Curated by ChEMBL | Assay Description Inhibition of human ERG tail current expressed in HEK293 cells after 5 mins by patch clamp assay | Bioorg Med Chem 24: 1619-36 (2016) Article DOI: 10.1016/j.bmc.2016.02.031 BindingDB Entry DOI: 10.7270/Q29P33JV | |||||||||||
More data for this Ligand-Target Pair |