Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50207236 (CHEMBL3946960) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.55E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Korea Institutes of Science and Technology (KIST) Curated by ChEMBL | Assay Description Inhibition of human ERG expressed in CHOK1 cells by whole-cell patch clamp method | Eur J Med Chem 123: 665-672 (2016) Article DOI: 10.1016/j.ejmech.2016.07.032 BindingDB Entry DOI: 10.7270/Q2ZK5JN6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Voltage-dependent T-type calcium channel subunit alpha-1H (Homo sapiens (Human)) | BDBM50207236 (CHEMBL3946960) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Korea Institutes of Science and Technology (KIST) Curated by ChEMBL | Assay Description Inhibition of Cav3.2 alpha1H (unknown origin) expressed in HEK293 cells by whole-cell patch clamp method | Eur J Med Chem 123: 665-672 (2016) Article DOI: 10.1016/j.ejmech.2016.07.032 BindingDB Entry DOI: 10.7270/Q2ZK5JN6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Voltage-dependent T-type calcium channel subunit alpha-1G (Homo sapiens (Human)) | BDBM50207236 (CHEMBL3946960) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Korea Institutes of Science and Technology (KIST) Curated by ChEMBL | Assay Description Inhibition of Cav3.1 alpha1G (unknown origin) expressed in HEK293 cells by whole-cell patch clamp method | Eur J Med Chem 123: 665-672 (2016) Article DOI: 10.1016/j.ejmech.2016.07.032 BindingDB Entry DOI: 10.7270/Q2ZK5JN6 | |||||||||||
More data for this Ligand-Target Pair |